# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5198038 | 24 | Drug metabolism | 0 | ALA5098722 | Metabolite_Notdetected | ||||||
2. | ALA5198038 | 24 | Drug metabolism | 0 | ALA5098721 | Metabolite_Notdetected | ||||||
3. | ALA5198038 | 24 | Drug metabolism | 0 | ALA5098720 | Metabolite_Notdetected | ||||||
4. | ALA5198038 | 24 | INH | = | 63 | % | ALA5098705 | % | Homo sapiens | |||
5. | ALA5198038 | 24 | INH | = | 71 | % | ALA5098700 | % | Homo sapiens | |||
6. | ALA5198038 | 24 | INH | = | 99 | % | ALA5098699 | % | Homo sapiens | |||
7. | ALA5198038 | 24 | CLH | < | 1 | uL/min | ALA5098696 | uL/min | ||||
8. | ALA5198038 | 24 | CLH | < | 3 | uL/min | ALA5098695 | uL/min | ||||
9. | ALA5198038 | 24 | CLH | = | 2.3 | uL/min | ALA5098694 | uL/min | ||||
10. | ALA5198038 | 24 | beta t1/2 | = | 1.7 | hr | ALA5098690 | hr | ||||
11. | ALA5198038 | 24 | CL | = | 77 | ml/min.kg | ALA5098689 | mL.min-1.kg-1 | ||||
12. | ALA5198038 | 24 | Vd | = | 5.9 | L/Kg | ALA5098688 | L.kg-1 | ||||
13. | ALA5198038 | 24 | pKa | = | 7.9 | ALA5098687 | ||||||
14. | ALA5198038 | 24 | IC50 | = | 2 | uM | ALA5098686 | 5.70 | nM | Homo sapiens | ||
15. | ALA5198038 | 24 | IC50 | = | 2.1 | uM | ALA5098682 | 5.68 | nM | Homo sapiens | ||
16. | ALA5198038 | 24 | INH | = | 11 | % | ALA5098681 | % | Homo sapiens | |||
17. | ALA5198038 | 24 | IC50 | = | 0.04 | uM | ALA5098680 | 7.40 | nM | Homo sapiens | ||
18. | ALA5198038 | 24 | IC50 | = | 0.46 | uM | ALA5098679 | 6.34 | nM | Homo sapiens | ||
19. | ALA5198038 | 24 | solubility | = | 110 | uM | ALA5098678 | nM | ||||
20. | ALA5198038 | 24 | logD | = | 1.9 | ALA5098677 |