# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5200047 | 12b | CLH | = | 69 | microL/min/mg | ALA5161361 | mL.min-1.g-1 | ||||
2. | ALA5200047 | 12b | t1/2 | = | 10 | min | ALA5161360 | hr | ||||
3. | ALA5200047 | 12b | Stability | = | 2 | % | ALA5161359 | % | ||||
4. | ALA5200047 | 12b | CLH | = | 78 | microL/min/mg | ALA5161358 | mL.min-1.g-1 | ||||
5. | ALA5200047 | 12b | t1/2 | = | 9 | min | ALA5161357 | hr | ||||
6. | ALA5200047 | 12b | Stability | = | 1 | % | ALA5161356 | % | ||||
7. | ALA5200047 | 12b | CLH | = | 19 | microL/min/mg | ALA5161355 | mL.min-1.g-1 | ||||
8. | ALA5200047 | 12b | t1/2 | = | 36 | min | ALA5161354 | hr | ||||
9. | ALA5200047 | 12b | Stability | = | 34 | % | ALA5161353 | % | ||||
10. | ALA5200047 | 12b | LD50 | > | 100 | uM | ALA5161352 | uM | Homo sapiens | |||
11. | ALA5200047 | 12b | Kinetic_solubility | = | 13.7 | uM | ALA5161351 | nM | ||||
12. | ALA5200047 | 12b | permeability | = | 9.1 | 10^-6 cm/s | ALA5161350 | 10^-6 cm/s | ||||
13. | ALA5200047 | 12b | IC50 | = | 4.01 | nM | ALA5161349 | 8.40 | nM | Mus musculus | ||
14. | ALA5200047 | 12b | IC50 | = | 15 | nM | ALA5161348 | 7.82 | nM | Mus musculus | ||
15. | ALA5200047 | 12b | IC50 | = | 416 | nM | ALA5161347 | 6.38 | nM | Homo sapiens | ||
16. | ALA5200047 | 12b | IC50 | = | 2.71 | nM | ALA5161346 | 8.57 | nM | Homo sapiens | ||
17. | ALA5200047 | 12b | IC50 | = | 1 | nM | ALA5161345 | 9.00 | nM | Homo sapiens |