| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5200108 | 47 | IC50 | > | 30 | uM | ALA5247304 | nM | Homo sapiens | |||
| 2. | ALA5200108 | 47 | IC50 | > | 20 | uM | ALA5247303 | nM | Homo sapiens | |||
| 3. | ALA5200108 | 47 | CLH | = | 48 | ml/min.kg | ALA5247302 | mL.min-1.kg-1 | ||||
| 4. | ALA5200108 | 47 | permeability | = | -4.5 | 10^-6 cm/s | ALA5247301 | 10^-6 cm/s | ||||
| 5. | ALA5200108 | 47 | logD | = | 3.9 | ALA5247300 | ||||||
| 6. | ALA5200108 | 47 | solubility | = | 0.03 | uM | ALA5247299 | nM | ||||
| 7. | ALA5200108 | 47 | solubility | = | 0.013 | uM | ALA5247298 | nM | ||||
| 8. | ALA5200108 | 47 | Cmax | = | 746 | nM | ALA5105222 | nM | ||||
| 9. | ALA5200108 | 47 | Tmax | = | 1.5 | hr | ALA5105221 | hr | ||||
| 10. | ALA5200108 | 47 | t1/2 | = | 11.6 | hr | ALA5105220 | hr | ||||
| 11. | ALA5200108 | 47 | AUC | = | 613 | nM.hr | ALA5105219 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 12. | ALA5200108 | 47 | CL | = | 23.7 | ml/min.kg | ALA5105218 | mL.min-1.kg-1 | ||||
| 13. | ALA5200108 | 47 | F | = | 29.3 | % | ALA5105183 | % | ||||
| 14. | ALA5200108 | 47 | IC50 | = | 87 | nM | ALA5105182 | 7.06 | nM | Homo sapiens |
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