# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5200341 | PROTAC 2 | Activity | 0 | ALA5113366 | Active | Homo sapiens | |||||
2. | ALA5200341 | PROTAC 2 | Activity | 0 | ALA5113361 | NA | Homo sapiens | |||||
3. | ALA5200341 | PROTAC 2 | Activity | 0 | ALA5113360 | NA | Homo sapiens | |||||
4. | ALA5200341 | PROTAC 2 | Activity | 0 | ALA5113359 | NA | Homo sapiens | |||||
5. | ALA5200341 | PROTAC 2 | Activity | 0 | ALA5113358 | Active | Homo sapiens | |||||
6. | ALA5200341 | PROTAC 2 | EC50 | = | 27.6 | pM | ALA5113357 | 10.56 | nM | Homo sapiens | ||
7. | ALA5200341 | PROTAC 2 | IC50 | = | 196.3 | nM | ALA5113356 | 6.71 | nM | Homo sapiens | ||
8. | ALA5200341 | PROTAC 2 | Stability | = | 80 | % | ALA5256462 | % | ||||
9. | ALA5200341 | PROTAC 2 | Stability | = | 93 | % | ALA5256461 | % | ||||
10. | ALA5200341 | PROTAC 2 | Papp | = | 0.049 | 10^-6 cm/s | ALA5256460 | 10^-6 cm/s | ||||
11. | ALA5200341 | PROTAC 2 | logD | = | 3.33 | ALA5256459 | ||||||
12. | ALA5200341 | PROTAC 2 | solubility | < | 0.5 | uM | ALA5256458 | nM | ||||
13. | ALA5200341 | PROTAC 2 | DC50 | = | 175 | pM | ALA5256457 | pM | Homo sapiens |