# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5200502 | 11 | Drug metabolism | 0 | ALA5149765 | Metabolite_Detected | ||||||
2. | ALA5200502 | 11 | Drugexcretion | = | 57 | % | ALA5149764 | % | ||||
3. | ALA5200502 | 11 | Papp | < | 0.2 | 10^-6 cm/s | ALA5149747 | 10^-6 cm/s | ||||
4. | ALA5200502 | 11 | INH | 0 | ALA5149746 | Dde | % | |||||
5. | ALA5200502 | 11 | Activity | = | 24 | % | ALA5149745 | % | ||||
6. | ALA5200502 | 11 | Activity | = | 56 | % | ALA5149744 | % | ||||
7. | ALA5200502 | 11 | Activity | = | 2 | ALA5149743 | ||||||
8. | ALA5200502 | 11 | AUC/dose | = | 6 | ng.hr/ml | ALA5149738 | ng.hr/ml | ||||
9. | ALA5200502 | 11 | Cmax | = | 6 | ng/ml | ALA5149737 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
10. | ALA5200502 | 11 | pIC50 | = | 7.6 | ALA5149727 | 7.60 | nM | Rattus norvegicus | |||
11. | ALA5200502 | 11 | pIC50 | = | 7.1 | ALA5149726 | 7.10 | nM | Homo sapiens |