# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | DS69910557 | 19e; DS69910557 | INH | < | 50 | % | ALA5148079 | % | ||||
2. | DS69910557 | 19e; DS69910557 | INH | < | 50 | % | ALA5148078 | % | Homo sapiens | |||
3. | DS69910557 | 19e; DS69910557 | INH | < | 50 | % | ALA5148077 | % | Homo sapiens | |||
4. | DS69910557 | 19e; DS69910557 | INH | < | 50 | % | ALA5148076 | % | ||||
5. | DS69910557 | 19e; DS69910557 | INH | < | 50 | % | ALA5148075 | % | Homo sapiens | |||
6. | DS69910557 | 19e; DS69910557 | INH | < | 50 | % | ALA5148074 | % | Homo sapiens | |||
7. | DS69910557 | 19e; DS69910557 | Activity | 0 | ALA5148073 | Active | ||||||
8. | DS69910557 | 19e; DS69910557 | logD | = | 2.2 | ALA5148072 | ||||||
9. | DS69910557 | 19e; DS69910557 | AUClast | = | 20.7 | hr.microg/ml | ALA5148071 | ng.hr.mL-1 | ||||
10. | DS69910557 | 19e; DS69910557 | Cmax | = | 1.42 | ug ml-1 | ALA5148070 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
11. | DS69910557 | 19e; DS69910557 | INH | = | 2 | % | ALA5148069 | % | Homo sapiens | |||
12. | DS69910557 | 19e; DS69910557 | solubility | = | 120 | ug ml-1 | ALA5148068 | ug.mL-1 | ||||
13. | DS69910557 | 19e; DS69910557 | solubility | = | 250 | ug ml-1 | ALA5148067 | ug.mL-1 | ||||
14. | DS69910557 | 19e; DS69910557 | Stability | = | 89 | % | ALA5148066 | % | ||||
15. | DS69910557 | 19e; DS69910557 | IC50 | = | 0.08 | uM | ALA5148065 | 7.10 | nM | Homo sapiens |