# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | [¹¹C]GSK215083 | [11C]142; [11C]GSK215083 | Ki | = | 0.16 | nM | ALA5110018 | 9.80 | nM | Homo sapiens | ||
2. | [¹¹C]GSK215083 | [11C]142; [11C]GSK215083 | Drug uptake | = | 11.5 | %Idose/L | ALA5110017 | %Idose/L | ||||
3. | [¹¹C]GSK215083 | [11C]142; [11C]GSK215083 | Drug uptake | = | 10.5 | %Idose/L | ALA5110016 | %Idose/L | ||||
4. | [¹¹C]GSK215083 | [11C]142; [11C]GSK215083 | Drug uptake | = | 3.5 | %Idose/L | ALA5110015 | %Idose/L | ||||
5. | [¹¹C]GSK215083 | [11C]142; [11C]GSK215083 | Ki | = | 0.79 | nM | ALA5110014 | 9.10 | nM | Homo sapiens |