| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5201690 | 21i | F | = | 44.9 | % | ALA5158011 | % | ||||
| 2. | ALA5201690 | 21i | Tmax | = | 2.3 | hr | ALA5158009 | hr | ||||
| 3. | ALA5201690 | 21i | Cmax | = | 1071.2 | ng/ml | ALA5158007 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 4. | ALA5201690 | 21i | Vdss | = | 2.6 | L/Kg | ALA5158005 | L.kg-1 | ||||
| 5. | ALA5201690 | 21i | CL | = | 13.1 | ml/min.kg | ALA5158004 | mL.min-1.kg-1 | ||||
| 6. | ALA5201690 | 21i | AUC | = | 5187.6 | ng.hr/ml | ALA5158002 | ng.hr.mL-1 | ||||
| 7. | ALA5201690 | 21i | AUC | = | 1155.5 | ng.hr/ml | ALA5158001 | ng.hr.mL-1 | ||||
| 8. | ALA5201690 | 21i | t1/2 | = | 3.1 | hr | ALA5157998 | hr | ||||
| 9. | ALA5201690 | 21i | t1/2 | = | 2.4 | hr | ALA5157997 | hr | ||||
| 10. | ALA5201690 | 21i | Stability | = | 95.1 | % | ALA5157994 | % | ||||
| 11. | ALA5201690 | 21i | Stability | = | 96.7 | % | ALA5157993 | % | ||||
| 12. | ALA5201690 | 21i | Stability | = | 93.8 | % | ALA5157992 | % | ||||
| 13. | ALA5201690 | 21i | INH | > | 99 | % | ALA5157991 | % | Homo sapiens | |||
| 14. | ALA5201690 | 21i | INH | > | 99 | % | ALA5157990 | % | Homo sapiens | |||
| 15. | ALA5201690 | 21i | INH | > | 99 | % | ALA5157989 | % | Homo sapiens | |||
| 16. | ALA5201690 | 21i | INH | = | 97.7 | % | ALA5157988 | % | Homo sapiens | |||
| 17. | ALA5201690 | 21i | INH | > | 99 | % | ALA5157987 | % | Homo sapiens | |||
| 18. | ALA5201690 | 21i | EC50 | > | 10000 | nM | ALA5157986 | nM | Homo sapiens | |||
| 19. | ALA5201690 | 21i | EC50 | = | 112 | nM | ALA5157985 | 6.95 | nM | Homo sapiens | ||
| 20. | ALA5201690 | 21i | EC50 | = | 34.6 | nM | ALA5157984 | 7.46 | nM | Homo sapiens |
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