| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  DS-3801b free base | 12 | INH | = | 3.1 | % | ALA5145236 | % | Homo sapiens | |||
| 2. | DS-3801b free base | 12 | INH | = | 8.8 | % | ALA5145235 | % | Homo sapiens | |||
| 3. | DS-3801b free base | 12 | INH | = | 5.3 | % | ALA5145234 | % | Homo sapiens | |||
| 4. | DS-3801b free base | 12 | INH | = | 13 | % | ALA5145233 | % | Homo sapiens | |||
| 5. | DS-3801b free base | 12 | PB | = | 66.5 | % | ALA5145232 | % | ||||
| 6. | DS-3801b free base | 12 | PB | = | 77.2 | % | ALA5145231 | % | ||||
| 7. | DS-3801b free base | 12 | Peff | = | 48 | 10^-6 cm/s | ALA5145230 | 10^-6 cm/s | ||||
| 8. | DS-3801b free base | 12 | Peff | = | 1.5 | 10^-6 cm/s | ALA5145229 | 10^-6 cm/s | ||||
| 9. | DS-3801b free base | 12 | Ratio EC50 | = | 11 | ALA5145228 | ||||||
| 10. | DS-3801b free base | 12 | EC50 | = | 7.3 | nM | ALA5145227 | 8.14 | nM | |||
| 11. | DS-3801b free base | 12 | logD | = | 1.3 | ALA5145226 | ||||||
| 12. | DS-3801b free base | 12 | Activity | = | 74 | % | ALA5145225 | % | Homo sapiens | |||
| 13. | DS-3801b free base | 12 | EC50 | = | 1.3 | nM | ALA5145224 | 8.89 | nM | |||
| 14. | DS-3801b free base | 12 | EC50 | = | 5.3 | nM | ALA5145222 | 8.28 | nM | Homo sapiens |
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