# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5202088 | 12f; EML980 | Activity | = | 80 | % | ALA5138969 | % | Homo sapiens | |||
2. | ALA5202088 | 12f; EML980 | Activity | 0 | ALA5138968 | Non-Toxic | Homo sapiens | |||||
3. | ALA5202088 | 12f; EML980 | permeability | 0 | ALA5138967 | Impermeable | ||||||
4. | ALA5202088 | 12f; EML980 | Time | = | 14.7 | s | ALA5138966 | hr | Homo sapiens | |||
5. | ALA5202088 | 12f; EML980 | K | = | 0.068 | 1/s | ALA5138965 | 1/s | Homo sapiens | |||
6. | ALA5202088 | 12f; EML980 | K | = | 2.7 | 10^6/Ms | ALA5138964 | 10^6/Ms | Homo sapiens | |||
7. | ALA5202088 | 12f; EML980 | Kd | = | 252 | nM | ALA5138963 | 6.60 | nM | Homo sapiens | ||
8. | ALA5202088 | 12f; EML980 | Selectivity Index | = | 619 | ALA5138956 | ||||||
9. | ALA5202088 | 12f; EML980 | Selectivity Index | = | 23 | ALA5138955 | ||||||
10. | ALA5202088 | 12f; EML980 | Selectivity Index | = | 2340 | ALA5138954 | ||||||
11. | ALA5202088 | 12f; EML980 | Selectivity Index | = | 12 | ALA5138953 | ||||||
12. | ALA5202088 | 12f; EML980 | Selectivity Index | = | 1082 | ALA5138952 | ||||||
13. | ALA5202088 | 12f; EML980 | Selectivity Index | = | 501 | ALA5138951 | ||||||
14. | ALA5202088 | 12f; EML980 | IC50 | = | 6 | uM | ALA5138950 | 5.22 | nM | Homo sapiens | ||
15. | ALA5202088 | 12f; EML980 | IC50 | = | 0.226 | uM | ALA5138949 | 6.65 | nM | Homo sapiens | ||
16. | ALA5202088 | 12f; EML980 | IC50 | = | 22.7 | uM | ALA5138948 | 4.64 | nM | Homo sapiens | ||
17. | ALA5202088 | 12f; EML980 | IC50 | = | 0.113 | uM | ALA5138947 | 6.95 | nM | Homo sapiens | ||
18. | ALA5202088 | 12f; EML980 | IC50 | = | 0.01 | uM | ALA5138946 | 8.01 | nM | Homo sapiens | ||
19. | ALA5202088 | 12f; EML980 | IC50 | = | 10.5 | uM | ALA5138945 | 4.98 | nM | Homo sapiens | ||
20. | ALA5202088 | 12f; EML980 | IC50 | = | 4.86 | uM | ALA5138944 | 5.31 | nM | Homo sapiens |