| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5202349 | 31 | Activity | 0 | ALA5155980 | NA | Mus musculus | |||||
| 2. | ALA5202349 | 31 | Ki | = | 17.6 | nM | ALA5155979 | 7.75 | nM | Mus musculus | ||
| 3. | ALA5202349 | 31 | Ki | = | 317 | nM | ALA5155978 | 6.50 | nM | Mus musculus | ||
| 4. | ALA5202349 | 31 | Activity | 0 | ALA5155977 | Active | Mus musculus | |||||
| 5. | ALA5202349 | 31 | t1/2 | = | 6.51 | min | ALA5155976 | hr | ||||
| 6. | ALA5202349 | 31 | t1/2 | = | 22.5 | min | ALA5155975 | hr | ||||
| 7. | ALA5202349 | 31 | t1/2 | = | 9.15 | min | ALA5155974 | hr | ||||
| 8. | ALA5202349 | 31 | Ratio | = | 48.9 | ALA5155973 | ||||||
| 9. | ALA5202349 | 31 | Papp | = | 0.51 | 10^-6 cm/s | ALA5155972 | 10^-6 cm/s | ||||
| 10. | ALA5202349 | 31 | Stability | = | 94.6 | % | ALA5155971 | % | ||||
| 11. | ALA5202349 | 31 | Stability | = | 84.6 | % | ALA5155970 | % | ||||
| 12. | ALA5202349 | 31 | Stability | = | 56.9 | % | ALA5155969 | % | ||||
| 13. | ALA5202349 | 31 | IC50 | = | 0.83 | uM | ALA5155968 | 6.08 | nM | Homo sapiens | ||
| 14. | ALA5202349 | 31 | IC50 | > | 30 | uM | ALA5155967 | nM | Homo sapiens | |||
| 15. | ALA5202349 | 31 | IC50 | > | 30 | uM | ALA5155966 | nM | Homo sapiens | |||
| 16. | ALA5202349 | 31 | IC50 | > | 30 | uM | ALA5155965 | nM | Homo sapiens | |||
| 17. | ALA5202349 | 31 | IC50 | = | 0.25 | uM | ALA5155964 | 6.60 | nM | Homo sapiens | ||
| 18. | ALA5202349 | 31 | Stability | = | 100 | % | ALA5155963 | % | ||||
| 19. | ALA5202349 | 31 | Stability | = | 64.5 | % | ALA5155962 | % | ||||
| 20. | ALA5202349 | 31 | Emax | = | 123 | % | ALA5155961 | % | Homo sapiens |
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