# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5202479 | TH-16 | IC50 | = | 2.244 | uM | ALA5142062 | 5.65 | nM | Homo sapiens | ||
2. | ALA5202479 | TH-16 | IC50 | = | 0.668 | uM | ALA5142061 | 6.17 | nM | Homo sapiens | ||
3. | ALA5202479 | TH-16 | IC50 | = | 0.53 | uM | ALA5142060 | 6.28 | nM | Homo sapiens | ||
4. | ALA5202479 | TH-16 | IC50 | = | 28.045 | uM | ALA5142059 | 4.55 | nM | Homo sapiens | ||
5. | ALA5202479 | TH-16 | IC50 | = | 16.508 | uM | ALA5142058 | 4.78 | nM | Homo sapiens | ||
6. | ALA5202479 | TH-16 | INH | = | 22 | % | ALA5142057 | % | Homo sapiens | |||
7. | ALA5202479 | TH-16 | INH | = | 71 | % | ALA5142056 | % | Homo sapiens | |||
8. | ALA5202479 | TH-16 | IC50 | = | 323 | nM | ALA5142055 | 6.49 | nM | Homo sapiens | ||
9. | ALA5202479 | TH-16 | IC50 | = | 105 | nM | ALA5142054 | 6.98 | nM | Homo sapiens | ||
10. | ALA5202479 | TH-16 | IC50 | = | 96 | nM | ALA5142053 | 7.02 | nM | Mus musculus | ||
11. | ALA5202479 | TH-16 | IC50 | = | 101 | nM | ALA5142052 | 7.00 | nM | Homo sapiens | ||
12. | ALA5202479 | TH-16 | IC50 | = | 77 | nM | ALA5142051 | 7.11 | nM | Homo sapiens | ||
13. | ALA5202479 | TH-16 | IC50 | = | 97 | nM | ALA5142050 | 7.01 | nM | Homo sapiens | ||
14. | ALA5202479 | TH-16 | IC50 | = | 0.114 | uM | ALA5142049 | 6.94 | nM | Homo sapiens |