| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5202526 | Q-c4 | K | = | 0.11 | /s | ALA5143809 | /s | Human immunodeficiency virus 1 | |||
| 2. | ALA5202526 | Q-c4 | IC50 | = | 3.47 | uM | ALA5143808 | 5.46 | nM | Human immunodeficiency virus 1 | ||
| 3. | ALA5202526 | Q-c4 | IC50 | = | 26.31 | uM | ALA5143807 | 4.58 | nM | Human immunodeficiency virus 1 | ||
| 4. | ALA5202526 | Q-c4 | Stability | = | 95 | % | ALA5143806 | % | ||||
| 5. | ALA5202526 | Q-c4 | Stability | = | 102.4 | % | ALA5143805 | % | ||||
| 6. | ALA5202526 | Q-c4 | Stability | = | 0 | % | ALA5143804 | % | ||||
| 7. | ALA5202526 | Q-c4 | CLH | = | 1799.6 | microL/min/mg | ALA5143803 | mL.min-1.g-1 | ||||
| 8. | ALA5202526 | Q-c4 | t1/2 | = | 0.8 | min | ALA5143802 | hr | ||||
| 9. | ALA5202526 | Q-c4 | Activity | = | 0.6 | % | ALA5143799 | % | Human immunodeficiency virus 1 | |||
| 10. | ALA5202526 | Q-c4 | Activity | = | 86.6 | % | ALA5143798 | % | Human immunodeficiency virus 1 | |||
| 11. | ALA5202526 | Q-c4 | Ratio | = | 0.86 | ALA5143797 | ||||||
| 12. | ALA5202526 | Q-c4 | Kd | = | 9.04 | uM | ALA5143796 | 5.04 | nM | Human immunodeficiency virus 1 | ||
| 13. | ALA5202526 | Q-c4 | Kd | = | 7.79 | uM | ALA5143795 | 5.11 | nM | Human immunodeficiency virus 1 | ||
| 14. | ALA5202526 | Q-c4 | Ratio CC50/EC50 | < | 1 | ALA5143794 | ||||||
| 15. | ALA5202526 | Q-c4 | Ratio CC50/EC50 | = | 25.49 | ALA5143793 | ||||||
| 16. | ALA5202526 | Q-c4 | CC50 | = | 14.53 | uM | ALA5143792 | nM | Homo sapiens | |||
| 17. | ALA5202526 | Q-c4 | EC50 | > | 14.53 | uM | ALA5143791 | nM | Human immunodeficiency virus 1 | |||
| 18. | ALA5202526 | Q-c4 | EC50 | = | 0.57 | uM | ALA5143790 | 6.24 | nM | Human immunodeficiency virus 1 | ||
| 19. | ALA5202526 | Q-c4 | CLH | = | 1619.6 | ml/min.kg | ALA5143789 | mL.min-1.kg-1 |
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