# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5202967 | KPH2f | IC50 | = | 3.14 | uM | ALA5157470 | 5.50 | nM | |||
2. | ALA5202967 | KPH2f | IC50 | = | 0.31 | uM | ALA5157469 | 6.51 | nM | |||
3. | ALA5202967 | KPH2f | IC50 | = | 0.78 | uM | ALA5157468 | 6.11 | nM | |||
4. | ALA5202967 | KPH2f | IC50 | = | 1.57 | uM | ALA5157467 | 5.80 | nM | |||
5. | ALA5202967 | KPH2f | IC50 | = | 2.17 | uM | ALA5157466 | 5.66 | nM | |||
6. | ALA5202967 | KPH2f | IC50 | = | 1.89 | uM | ALA5157465 | 5.72 | nM | |||
7. | ALA5202967 | KPH2f | Activity | 0 | ALA5157464 | Non-Toxic | ||||||
8. | ALA5202967 | KPH2f | Activity | 0 | ALA5157463 | Non-Toxic | ||||||
9. | ALA5202967 | KPH2f | IC50 | = | 9.37 | uM | ALA5157462 | 5.03 | nM | Homo sapiens | ||
10. | ALA5202967 | KPH2f | IC50 | = | 167.24 | uM | ALA5157461 | nM | Homo sapiens | |||
11. | ALA5202967 | KPH2f | IC50 | = | 207.56 | uM | ALA5157460 | nM | Homo sapiens | |||
12. | ALA5202967 | KPH2f | F | = | 30.13 | % | ALA5157459 | % | ||||
13. | ALA5202967 | KPH2f | MRT | = | 4.8 | hr | ALA5157458 | hr | ||||
14. | ALA5202967 | KPH2f | MRT | = | 3.17 | hr | ALA5157457 | hr | ||||
15. | ALA5202967 | KPH2f | AUC | = | 18535.9 | ng/mL.hr | ALA5157456 | ng.hr.mL-1 | ||||
16. | ALA5202967 | KPH2f | AUC | = | 5656.03 | ng/mL.hr | ALA5157455 | ng.hr.mL-1 | ||||
17. | ALA5202967 | KPH2f | t1/2 | = | 4.19 | hr | ALA5157454 | hr | ||||
18. | ALA5202967 | KPH2f | t1/2 | = | 5.14 | hr | ALA5157453 | hr | ||||
19. | ALA5202967 | KPH2f | Cmax | = | 7649.04 | ng/ml | ALA5157452 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
20. | ALA5202967 | KPH2f | Tmax | = | 0.17 | hr | ALA5157451 | hr |