# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | LJ-4517 | 2; LJ-4517 | FC | = | 4.8 | ALA5130207 | Homo sapiens | |||||
2. | LJ-4517 | 2; LJ-4517 | FC | = | 26.2 | ALA5130206 | Homo sapiens | |||||
3. | LJ-4517 | 2; LJ-4517 | FC | = | 25 | ALA5130205 | Homo sapiens | |||||
4. | LJ-4517 | 2; LJ-4517 | FC | = | 28.6 | ALA5130204 | Homo sapiens | |||||
5. | LJ-4517 | 2; LJ-4517 | EC50 | = | 8390 | nM | ALA5130203 | 5.08 | nM | Homo sapiens | ||
6. | LJ-4517 | 2; LJ-4517 | EC50 | = | 109 | nM | ALA5130202 | 6.96 | nM | Homo sapiens | ||
7. | LJ-4517 | 2; LJ-4517 | EC50 | = | 94 | nM | ALA5130201 | 7.03 | nM | Homo sapiens | ||
8. | LJ-4517 | 2; LJ-4517 | EC50 | = | 0.9 | nM | ALA5130200 | 9.05 | nM | Homo sapiens | ||
9. | LJ-4517 | 2; LJ-4517 | Ki | = | 56.4 | nM | ALA5130199 | 7.25 | nM | Homo sapiens | ||
10. | LJ-4517 | 2; LJ-4517 | Ki | = | 19 | nM | ALA5130198 | 7.72 | nM | Homo sapiens | ||
11. | LJ-4517 | 2; LJ-4517 | Ki | = | 21.6 | nM | ALA5130197 | 7.67 | nM | Homo sapiens | ||
12. | LJ-4517 | 2; LJ-4517 | Ki | = | 18.3 | nM | ALA5130196 | 7.74 | nM | Homo sapiens | ||
13. | LJ-4517 | 2; LJ-4517 | Bmax | = | 2.1 | pmol | ALA5130195 | pmol | Homo sapiens | |||
14. | LJ-4517 | 2; LJ-4517 | Bmax | = | 2.4 | pmol | ALA5130194 | pmol | Homo sapiens | |||
15. | LJ-4517 | 2; LJ-4517 | Bmax | = | 2.2 | pmol | ALA5130193 | pmol | Homo sapiens | |||
16. | LJ-4517 | 2; LJ-4517 | Bmax | = | 2.03 | pmol | ALA5130192 | pmol | Homo sapiens | |||
17. | LJ-4517 | 2; LJ-4517 | Kd | = | 2.7 | nM | ALA5130191 | 8.57 | nM | Homo sapiens | ||
18. | LJ-4517 | 2; LJ-4517 | Kd | = | 2.9 | nM | ALA5130190 | 8.54 | nM | Homo sapiens | ||
19. | LJ-4517 | 2; LJ-4517 | Kd | = | 1.8 | nM | ALA5130189 | 8.74 | nM | Homo sapiens | ||
20. | LJ-4517 | 2; LJ-4517 | Kd | = | 1.95 | nM | ALA5130188 | 8.71 | nM | Homo sapiens |