# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5203787 | 21 | Activity | 0 | ALA5112607 | Dde | Mus musculus | |||||
2. | ALA5203787 | 21 | Activity | 0 | ALA5112606 | Active | Mus musculus | |||||
3. | ALA5203787 | 21 | Activity | 0 | ALA5112605 | Dde | Mus musculus | |||||
4. | ALA5203787 | 21 | Activity | 0 | ALA5112604 | Active | Mus musculus | |||||
5. | ALA5203787 | 21 | Activity | 0 | ALA5112602 | Dde | Mus musculus | |||||
6. | ALA5203787 | 21 | AUC | = | 13.6 | microg.hr/mL | ALA5112597 | ng.hr.mL-1 | ||||
7. | ALA5203787 | 21 | AUClast | = | 13.5 | microg.hr/mL | ALA5112596 | ng.hr.mL-1 | ||||
8. | ALA5203787 | 21 | Cmax | = | 19.1 | ug ml-1 | ALA5112595 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
9. | ALA5203787 | 21 | Tmax | = | 0.25 | hr | ALA5112594 | hr | ||||
10. | ALA5203787 | 21 | t1/2 | = | 0.7 | hr | ALA5112593 | hr | ||||
11. | ALA5203787 | 21 | IC50 | > | 10 | uM | ALA5112592 | nM | Homo sapiens | |||
12. | ALA5203787 | 21 | IC50 | > | 100 | uM | ALA5112591 | nM | Homo sapiens | |||
13. | ALA5203787 | 21 | INH | = | 2 | % | ALA5112590 | % | Homo sapiens | |||
14. | ALA5203787 | 21 | Ratio | = | 9.2 | ALA5112589 | ||||||
15. | ALA5203787 | 21 | Papp | = | 301.7 | nm/s | ALA5112588 | nm/s | ||||
16. | ALA5203787 | 21 | Papp | = | 32.9 | nm/s | ALA5112587 | nm/s | ||||
17. | ALA5203787 | 21 | INH | = | 2 | % | ALA5112584 | % | ||||
18. | ALA5203787 | 21 | INH | = | 32 | % | ALA5112582 | % | Homo sapiens | |||
19. | ALA5203787 | 21 | INH | = | 30 | % | ALA5112581 | % | Homo sapiens | |||
20. | ALA5203787 | 21 | LD50 | > | 100 | uM | ALA5112580 | uM | Homo sapiens |