# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5204021 | 27b; VU6019650 | IC50 | > | 5000 | nM | ALA5216737 | nM | Homo sapiens | |||
2. | ALA5204021 | 27b; VU6019650 | IC50 | > | 5000 | nM | ALA5216736 | nM | Homo sapiens | |||
3. | ALA5204021 | 27b; VU6019650 | IC50 | > | 10000 | nM | ALA5216735 | nM | Homo sapiens | |||
4. | ALA5204021 | 27b; VU6019650 | IC50 | = | 36 | nM | ALA5216718 | 7.44 | nM | Homo sapiens | ||
5. | ALA5204021 | 27b; VU6019650 | IC50 | > | 10000 | nM | ALA5216717 | nM | Homo sapiens | |||
6. | ALA5204021 | 27b; VU6019650 | Activity | = | 57.4 | % | ALA5164559 | % | Rattus norvegicus | |||
7. | ALA5204021 | 27b; VU6019650 | Activity | = | 31.7 | % | ALA5164558 | % | Rattus norvegicus | |||
8. | ALA5204021 | 27b; VU6019650 | Activity | = | 18.9 | % | ALA5164557 | % | Rattus norvegicus | |||
9. | ALA5204021 | 27b; VU6019650 | Papp | = | 26.8 | 10^-6 cm/s | ALA5164556 | 10^-6 cm/s | ||||
10. | ALA5204021 | 27b; VU6019650 | Ratio | = | 2.85 | ALA5164555 | ||||||
11. | ALA5204021 | 27b; VU6019650 | Activity | = | 3.57 | Hz | ALA5164554 | Hz | ||||
12. | ALA5204021 | 27b; VU6019650 | Activity | = | 3.07 | Hz | ALA5164553 | Hz | ||||
13. | ALA5204021 | 27b; VU6019650 | Activity | = | 3.22 | Hz | ALA5164553 | Hz | ||||
14. | ALA5204021 | 27b; VU6019650 | IC50 | = | 125 | nM | ALA5164552 | 6.90 | nM | Rattus norvegicus | ||
15. | ALA5204021 | 27b; VU6019650 | IC50 | = | 2.2 | nM | ALA5164551 | 8.66 | nM | Rattus norvegicus | ||
16. | ALA5204021 | 27b; VU6019650 | Activity | 0 | ALA5164550 | Active | Rattus norvegicus | |||||
17. | ALA5204021 | 27b; VU6019650 | Ki | = | 68 | nM | ALA5164549 | 7.17 | nM | Rattus norvegicus | ||
18. | ALA5204021 | 27b; VU6019650 | F | = | 27.6 | % | ALA5164548 | % | ||||
19. | ALA5204021 | 27b; VU6019650 | AUC | = | 830 | hr.ng/ml | ALA5164547 | ng.hr.mL-1 | ||||
20. | ALA5204021 | 27b; VU6019650 | Tmax | = | 0.25 | hr | ALA5164546 | hr |