# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5204493 | 15h | CL | = | 7.99 | ml/min.kg | ALA5148242 | mL.min-1.kg-1 | ||||
2. | ALA5204493 | 15h | Kp | = | 0.67 | ALA5148241 | ||||||
3. | ALA5204493 | 15h | Kp | = | 3.34 | ALA5148240 | ||||||
4. | ALA5204493 | 15h | Cmax | = | 43 | ng/ml | ALA5148239 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
5. | ALA5204493 | 15h | AUC | = | 251 | ng.hr/ml | ALA5148238 | ng.hr.mL-1 | ||||
6. | ALA5204493 | 15h | Stability | = | 86 | % | ALA5148237 | % | ||||
7. | ALA5204493 | 15h | Stability | = | 98 | % | ALA5148236 | % | ||||
8. | ALA5204493 | 15h | IC50 | = | 3.7 | uM | ALA5148231 | 5.43 | nM | Homo sapiens | ||
9. | ALA5204493 | 15h | Fu | = | 1 | % | ALA5148230 | |||||
10. | ALA5204493 | 15h | EC150 | = | 0.002 | uM | ALA5148229 | uM | Homo sapiens |