# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5204764 | 11a | Fu | = | 1.5 | % | ALA5250297 | |||||
2. | ALA5204764 | 11a | Ki | > | 10000 | nM | ALA5250282 | nM | Homo sapiens | |||
3. | ALA5204764 | 11a | Fu | = | 0.3 | % | ALA5250281 | |||||
4. | ALA5204764 | 11a | CLH | = | 287.1 | ml/min.kg | ALA5250280 | mL.min-1.kg-1 | ||||
5. | ALA5204764 | 11a | CLH | = | 144.7 | ml/min.kg | ALA5250279 | mL.min-1.kg-1 | ||||
6. | ALA5204764 | 11a | Ki | > | 10000 | nM | ALA5250278 | nM | Homo sapiens | |||
7. | ALA5204764 | 11a | Ki | = | 2463 | nM | ALA5250277 | 5.61 | nM | Homo sapiens | ||
8. | ALA5204764 | 11a | Ki | = | 299 | nM | ALA5250275 | 6.52 | nM | Homo sapiens | ||
9. | ALA5204764 | 11a | pKi | = | 6.52 | ALA5250271 | 6.52 | nM | Homo sapiens | |||
10. | ALA5204764 | 11a | Ki | = | 299 | nM | ALA5250271 | 6.52 | nM | Homo sapiens | ||
11. | ALA5204764 | 11a | pKi | = | 6.88 | ALA5250270 | 6.88 | nM | Homo sapiens | |||
12. | ALA5204764 | 11a | Ki | = | 131 | nM | ALA5250270 | 6.88 | nM | Homo sapiens | ||
13. | ALA5204764 | 11a | BPR | = | 2.9 | ALA5145681 | ||||||
14. | ALA5204764 | 11a | Drug uptake | = | 134 | ng/g | ALA5145680 | ng/g | ||||
15. | ALA5204764 | 11a | Cp | = | 45.8 | ng/ml | ALA5145679 | ng/ml | ||||
16. | ALA5204764 | 11a | AUC | = | 747 | hr.ng/ml | ALA5145678 | ng.hr.mL-1 | ||||
17. | ALA5204764 | 11a | Vdss | = | 5.5 | L/Kg | ALA5145677 | L.kg-1 | ||||
18. | ALA5204764 | 11a | C0 | = | 5.5 | ng/ml | ALA5145676 | ng/ml | ||||
19. | ALA5204764 | 11a | t1/2 | = | 4.4 | hr | ALA5145675 | hr | ||||
20. | ALA5204764 | 11a | CL | = | 22 | ml/min.kg | ALA5145674 | mL.min-1.kg-1 |