# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5204900 | 12a | CLH | = | 56 | microL/min/mg | ALA5161361 | mL.min-1.g-1 | ||||
2. | ALA5204900 | 12a | t1/2 | = | 12 | min | ALA5161360 | hr | ||||
3. | ALA5204900 | 12a | Stability | = | 4 | % | ALA5161359 | % | ||||
4. | ALA5204900 | 12a | CLH | = | 109 | microL/min/mg | ALA5161358 | mL.min-1.g-1 | ||||
5. | ALA5204900 | 12a | t1/2 | = | 6 | min | ALA5161357 | hr | ||||
6. | ALA5204900 | 12a | Stability | = | 1 | % | ALA5161356 | % | ||||
7. | ALA5204900 | 12a | CLH | = | 57 | microL/min/mg | ALA5161355 | mL.min-1.g-1 | ||||
8. | ALA5204900 | 12a | t1/2 | = | 12 | min | ALA5161354 | hr | ||||
9. | ALA5204900 | 12a | Stability | = | 4 | % | ALA5161353 | % | ||||
10. | ALA5204900 | 12a | LD50 | = | 92.8 | uM | ALA5161352 | uM | Homo sapiens | |||
11. | ALA5204900 | 12a | Kinetic_solubility | = | 42.6 | uM | ALA5161351 | nM | ||||
12. | ALA5204900 | 12a | permeability | = | 9.2 | 10^-6 cm/s | ALA5161350 | 10^-6 cm/s | ||||
13. | ALA5204900 | 12a | IC50 | = | 35.4 | nM | ALA5161349 | 7.45 | nM | Mus musculus | ||
14. | ALA5204900 | 12a | IC50 | = | 12.1 | nM | ALA5161348 | 7.92 | nM | Mus musculus | ||
15. | ALA5204900 | 12a | IC50 | = | 947 | nM | ALA5161347 | 6.02 | nM | Homo sapiens | ||
16. | ALA5204900 | 12a | IC50 | = | 14.5 | nM | ALA5161346 | 7.84 | nM | Homo sapiens | ||
17. | ALA5204900 | 12a | IC50 | = | 0.4 | nM | ALA5161345 | 9.40 | nM | Homo sapiens |