# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5206272 | 12c; EML736 | Time | = | 76.9 | s | ALA5138966 | hr | Homo sapiens | |||
2. | ALA5206272 | 12c; EML736 | K | = | 0.013 | 1/s | ALA5138965 | 1/s | Homo sapiens | |||
3. | ALA5206272 | 12c; EML736 | K | = | 3.49 | 10^4/Ms | ALA5138964 | 10^4/Ms | Homo sapiens | |||
4. | ALA5206272 | 12c; EML736 | Kd | = | 359.2 | nM | ALA5138963 | 6.45 | nM | Homo sapiens | ||
5. | ALA5206272 | 12c; EML736 | Selectivity Index | = | 14 | ALA5138956 | ||||||
6. | ALA5206272 | 12c; EML736 | Selectivity Index | = | 0.52 | ALA5138955 | ||||||
7. | ALA5206272 | 12c; EML736 | Selectivity Index | > | 238 | ALA5138954 | ||||||
8. | ALA5206272 | 12c; EML736 | Selectivity Index | = | 122 | ALA5138953 | ||||||
9. | ALA5206272 | 12c; EML736 | Selectivity Index | = | 51 | ALA5138952 | ||||||
10. | ALA5206272 | 12c; EML736 | Selectivity Index | = | 20 | ALA5138951 | ||||||
11. | ALA5206272 | 12c; EML736 | IC50 | = | 5.87 | uM | ALA5138950 | 5.23 | nM | Homo sapiens | ||
12. | ALA5206272 | 12c; EML736 | IC50 | = | 0.22 | uM | ALA5138949 | 6.66 | nM | Homo sapiens | ||
13. | ALA5206272 | 12c; EML736 | IC50 | > | 100 | uM | ALA5138948 | nM | Homo sapiens | |||
14. | ALA5206272 | 12c; EML736 | IC50 | = | 51.41 | uM | ALA5138947 | 4.29 | nM | Homo sapiens | ||
15. | ALA5206272 | 12c; EML736 | IC50 | = | 0.42 | uM | ALA5138946 | 6.38 | nM | Homo sapiens | ||
16. | ALA5206272 | 12c; EML736 | IC50 | = | 21.26 | uM | ALA5138945 | 4.67 | nM | Homo sapiens | ||
17. | ALA5206272 | 12c; EML736 | IC50 | = | 8.46 | uM | ALA5138944 | 5.07 | nM | Homo sapiens | ||
18. | ALA5206272 | 12c; EML736 | Activity | = | 0.3 | % | ALA5138942 | % | Homo sapiens |