| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5206328 | 1c | Drug uptake | = | 9.6 | % | ALA5167072 | % | ||||
| 2. | ALA5206328 | 1c | beta t1/2 | > | 24 | hr | ALA5167071 | hr | ||||
| 3. | ALA5206328 | 1c | Drug uptake | = | 8.4 | % | ALA5167070 | % | ||||
| 4. | ALA5206328 | 1c | Ratio | = | 149 | ALA5167069 | ||||||
| 5. | ALA5206328 | 1c | Ct | = | 29.8 | uM | ALA5167068 | uM | ||||
| 6. | ALA5206328 | 1c | Cmax | = | 1.08 | uM | ALA5167067 | nM | ||||
| 7. | ALA5206328 | 1c | Cmax | = | 0.09 | uM | ALA5167066 | nM | ||||
| 8. | ALA5206328 | 1c | INH | = | -3 | % | ALA5167065 | % | Rattus norvegicus | |||
| 9. | ALA5206328 | 1c | INH | = | 50 | % | ALA5167064 | % | Rattus norvegicus | |||
| 10. | ALA5206328 | 1c | PB | = | 99.6 | % | ALA5167063 | % | ||||
| 11. | ALA5206328 | 1c | PPB | > | 99.9 | % | ALA5167062 | % | ||||
| 12. | ALA5206328 | 1c | PPB | = | 99.9 | % | ALA5167061 | % | ||||
| 13. | ALA5206328 | 1c | permeability | = | 2.8 | 10^-6 cm/s | ALA5167060 | 10^-6 cm/s | ||||
| 14. | ALA5206328 | 1c | solubility | = | 0.01 | mg/ml | ALA5167059 | ug.mL-1 | ||||
| 15. | ALA5206328 | 1c | IC50 | > | 5000 | nM | ALA5167058 | nM | Homo sapiens | |||
| 16. | ALA5206328 | 1c | IC50 | = | 164 | nM | ALA5167057 | 6.79 | nM | Homo sapiens | ||
| 17. | ALA5206328 | 1c | IC50 | = | 0.2 | nM | ALA5167056 | 9.70 | nM | Homo sapiens | ||
| 18. | ALA5206328 | 1c | t1/2 | > | 16 | hr | ALA5167055 | hr | Homo sapiens | |||
| 19. | ALA5206328 | 1c | IC50 | = | 0.1 | nM | ALA5167054 | 10.00 | nM | |||
| 20. | ALA5206328 | 1c | IC50 | = | 0.2 | nM | ALA5167053 | 9.70 | nM | Homo sapiens |
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