# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5207561 | F2 | F | = | 63.71 | % | ALA5106052 | % | ||||
2. | ALA5207561 | F2 | Vd | = | 996 | ml/kg | ALA5106051 | L.kg-1 | ||||
3. | ALA5207561 | F2 | CL | = | 1190 | ml/hr/kg | ALA5106050 | mL.min-1.kg-1 | ||||
4. | ALA5207561 | F2 | AUC | = | 851 | hr.ng/ml | ALA5106049 | ng.hr.mL-1 | ||||
5. | ALA5207561 | F2 | AUCt | = | 847 | hr.ng/ml | ALA5106048 | ng.hr.mL-1 | ||||
6. | ALA5207561 | F2 | Cmax | = | 1933 | ng/ml | ALA5106047 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
7. | ALA5207561 | F2 | Tmax | = | 0.1 | hr | ALA5106046 | hr | ||||
8. | ALA5207561 | F2 | beta t1/2 | = | 0.57 | hr | ALA5106045 | hr | ||||
9. | ALA5207561 | F2 | AUC | = | 1637 | hr.ng/ml | ALA5106044 | ng.hr.mL-1 | ||||
10. | ALA5207561 | F2 | AUCt | = | 1619 | hr.ng/ml | ALA5106043 | ng.hr.mL-1 | ||||
11. | ALA5207561 | F2 | Cmax | = | 1026 | ng/ml | ALA5106042 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
12. | ALA5207561 | F2 | Tmax | = | 0.139 | hr | ALA5106041 | hr | ||||
13. | ALA5207561 | F2 | beta t1/2 | = | 1.32 | hr | ALA5106040 | hr | ||||
14. | ALA5207561 | F2 | Activity | = | 34.38 | uM | ALA5106039 | uM | Mus musculus | |||
15. | ALA5207561 | F2 | Activity | = | 30.48 | mg/dl | ALA5106038 | mg/dl | Mus musculus | |||
16. | ALA5207561 | F2 | Activity | = | 8.557 | uM | ALA5106037 | uM | Mus musculus | |||
17. | ALA5207561 | F2 | Activity | = | 29.23 | U/L | ALA5106036 | U/L | Mus musculus | |||
18. | ALA5207561 | F2 | Activity | = | 295 | uM | ALA5106035 | uM | Mus musculus | |||
19. | ALA5207561 | F2 | CC50 | = | 14.4 | uM | ALA5106034 | nM | Homo sapiens | |||
20. | ALA5207561 | F2 | INH | = | 84.48 | % | ALA5106033 | % | Homo sapiens |