# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5207564 | 73; BAY-1143269 | T/C | = | 0.33 | ALA5137674 | ||||||
2. | ALA5207564 | 73; BAY-1143269 | F | = | 78 | % | ALA5137673 | % | ||||
3. | ALA5207564 | 73; BAY-1143269 | F | = | 71 | % | ALA5137672 | % | ||||
4. | ALA5207564 | 73; BAY-1143269 | beta t1/2 | = | 1.2 | hr | ALA5137671 | hr | ||||
5. | ALA5207564 | 73; BAY-1143269 | beta t1/2 | = | 1.2 | hr | ALA5137670 | hr | ||||
6. | ALA5207564 | 73; BAY-1143269 | CL | = | 2.34 | L/Kg.hr | ALA5137669 | L/Kg.hr | ||||
7. | ALA5207564 | 73; BAY-1143269 | CL | = | 0.41 | L/Kg.hr | ALA5137668 | L/Kg.hr | ||||
8. | ALA5207564 | 73; BAY-1143269 | Vdss | = | 6 | L/Kg | ALA5137667 | L.kg-1 | ||||
9. | ALA5207564 | 73; BAY-1143269 | Vdss | = | 0.87 | L/Kg | ALA5137666 | L.kg-1 | ||||
10. | ALA5207564 | 73; BAY-1143269 | IC50 | = | 40 | nM | ALA5137665 | 7.40 | nM | Homo sapiens |