# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5207946 | PROTAC 4 | Activity | 0 | ALA5113366 | Active | Homo sapiens | |||||
2. | ALA5207946 | PROTAC 4 | Activity | 0 | ALA5113365 | NA | Homo sapiens | |||||
3. | ALA5207946 | PROTAC 4 | Activity | 0 | ALA5113364 | NA | Homo sapiens | |||||
4. | ALA5207946 | PROTAC 4 | Activity | 0 | ALA5113363 | NA | Homo sapiens | |||||
5. | ALA5207946 | PROTAC 4 | EC50 | = | 23.8 | pM | ALA5113357 | 10.62 | nM | Homo sapiens | ||
6. | ALA5207946 | PROTAC 4 | IC50 | = | 123.9 | nM | ALA5113356 | 6.91 | nM | Homo sapiens | ||
7. | ALA5207946 | PROTAC 4 | Stability | = | 72 | % | ALA5256462 | % | ||||
8. | ALA5207946 | PROTAC 4 | Stability | = | 90 | % | ALA5256461 | % | ||||
9. | ALA5207946 | PROTAC 4 | Papp | = | 0.009 | 10^-6 cm/s | ALA5256460 | 10^-6 cm/s | ||||
10. | ALA5207946 | PROTAC 4 | logD | = | 2.65 | ALA5256459 | ||||||
11. | ALA5207946 | PROTAC 4 | solubility | = | 2.91 | uM | ALA5256458 | nM | ||||
12. | ALA5207946 | PROTAC 4 | DC50 | = | 20 | pM | ALA5256457 | pM | Homo sapiens |