# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5207990 | 72 | EC50 | = | 77 | uM | ALA5158948 | 4.11 | nM | |||
2. | ALA5207990 | 72 | Ratio | = | 1.3 | ALA5158947 | ||||||
3. | ALA5207990 | 72 | Papp | = | 2.8 | 10^-6 cm/s | ALA5158946 | 10^-6 cm/s | ||||
4. | ALA5207990 | 72 | Papp | = | 2.2 | 10^-6 cm/s | ALA5158945 | 10^-6 cm/s | ||||
5. | ALA5207990 | 72 | Ratio | = | 61.7 | ALA5158944 | ||||||
6. | ALA5207990 | 72 | Papp | = | 18.2 | 10^-6 cm/s | ALA5158943 | 10^-6 cm/s | ||||
7. | ALA5207990 | 72 | Papp | = | 0.29 | 10^-6 cm/s | ALA5158942 | 10^-6 cm/s | ||||
8. | ALA5207990 | 72 | log Pe | = | 5.44 | ALA5158941 | ||||||
9. | ALA5207990 | 72 | Drug recovery | = | 86 | % | ALA5158940 | % | ||||
10. | ALA5207990 | 72 | PPB | = | 84 | % | ALA5158939 | % | ||||
11. | ALA5207990 | 72 | CLH | = | 2.37 | uL/min | ALA5158938 | uL/min | ||||
12. | ALA5207990 | 72 | t1/2 | = | 584 | min | ALA5158937 | hr | ||||
13. | ALA5207990 | 72 | t1/2 | = | 1075 | min | ALA5158936 | hr | ||||
14. | ALA5207990 | 72 | INH | 0 | ALA5158935 | NA | % | Homo sapiens | ||||
15. | ALA5207990 | 72 | INH | 0 | ALA5158934 | NA | % | Homo sapiens | ||||
16. | ALA5207990 | 72 | INH | 0 | ALA5158933 | NA | % | Homo sapiens | ||||
17. | ALA5207990 | 72 | INH | 0 | ALA5158932 | NA | % | Homo sapiens | ||||
18. | ALA5207990 | 72 | INH | 0 | ALA5158931 | Active | % | Homo sapiens | ||||
19. | ALA5207990 | 72 | Kinact | = | 0.46 | /min | ALA5158930 | /min | Homo sapiens | |||
20. | ALA5207990 | 72 | Ki | = | 1 | uM | ALA5158930 | 6.00 | nM | Homo sapiens |