| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  PA 8 | PA-8 | Activity | 0 | ALA5135039 | Active | Mus musculus | |||||
| 2. | PA 8 | PA-8 | t1/2 | = | 1.72 | hr | ALA5135038 | hr | ||||
| 3. | PA 8 | PA-8 | t1/2 | = | 2.19 | hr | ALA5135037 | hr | ||||
| 4. | PA 8 | PA-8 | Tmax | = | 0.5 | hr | ALA5135036 | hr | ||||
| 5. | PA 8 | PA-8 | Tmax | = | 0.67 | hr | ALA5135035 | hr | ||||
| 6. | PA 8 | PA-8 | Cmax | = | 0.79 | uM | ALA5135034 | nM | ||||
| 7. | PA 8 | PA-8 | Cmax | = | 14.35 | uM | ALA5135033 | nM | ||||
| 8. | PA 8 | PA-8 | PPB | = | 49.5 | % | ALA5135032 | % | ||||
| 9. | PA 8 | PA-8 | PPB | = | 69.6 | % | ALA5135031 | % | ||||
| 10. | PA 8 | PA-8 | Stability | = | 94 | % | ALA5135030 | % | ||||
| 11. | PA 8 | PA-8 | Stability | = | 91 | % | ALA5135029 | % | ||||
| 12. | PA 8 | PA-8 | Stability | = | 96 | % | ALA5135028 | % | ||||
| 13. | PA 8 | PA-8 | Stability | = | 93 | % | ALA5135027 | % | ||||
| 14. | PA 8 | PA-8 | permeability | = | 0.3 | 10^-6 cm/s | ALA5135026 | 10^-6 cm/s | ||||
| 15. | PA 8 | PA-8 | solubility | = | 92.2 | uM | ALA5135025 | nM | ||||
| 16. | PA 8 | PA-8 | Activity | 0 | ALA5135024 | Active | Mus musculus | |||||
| 17. | PA 8 | PA-8 | Activity | 0 | ALA5135023 | Active | Mus musculus | |||||
| 18. | PA 8 | PA-8 | Activity | 0 | ALA5135022 | Active | Mus musculus | |||||
| 19. | PA 8 | PA-8 | Activity | 0 | ALA5135018 | Dde | Homo sapiens | |||||
| 20. | PA 8 | PA-8 | IC50 | = | 1.48 | nM | ALA5135018 | 8.83 | nM | Homo sapiens |
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