# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5218639 | (rac)-30a; VU6029053 | Papp | = | 0.431 | 10^-6 cm/s | ALA5216734 | 10^-6 cm/s | ||||
2. | ALA5218639 | (rac)-30a; VU6029053 | Ratio | = | 110 | ALA5216733 | ||||||
3. | ALA5218639 | (rac)-30a; VU6029053 | Fu | = | 0.17 | ALA5216729 | ||||||
4. | ALA5218639 | (rac)-30a; VU6029053 | Fu | = | 0.26 | ALA5216728 | ||||||
5. | ALA5218639 | (rac)-30a; VU6029053 | Fu | = | 0.02 | ALA5216727 | ||||||
6. | ALA5218639 | (rac)-30a; VU6029053 | Activity | = | 51 | % | ALA5216726 | % | Homo sapiens | |||
7. | ALA5218639 | (rac)-30a; VU6029053 | IC50 | > | 10000 | nM | ALA5216725 | nM | Homo sapiens | |||
8. | ALA5218639 | (rac)-30a; VU6029053 | Activity | = | 3 | % | ALA5216723 | % | Rattus norvegicus | |||
9. | ALA5218639 | (rac)-30a; VU6029053 | IC50 | = | 572 | nM | ALA5216722 | 6.24 | nM | Rattus norvegicus | ||
10. | ALA5218639 | (rac)-30a; VU6029053 | CL | = | 260 | ml/min.kg | ALA5216721 | mL.min-1.kg-1 | ||||
11. | ALA5218639 | (rac)-30a; VU6029053 | CL | = | 7 | ml/min.kg | ALA5216720 | mL.min-1.kg-1 | ||||
12. | ALA5218639 | (rac)-30a; VU6029053 | Activity | = | 3 | % | ALA5216719 | % | Homo sapiens | |||
13. | ALA5218639 | (rac)-30a; VU6029053 | IC50 | = | 309 | nM | ALA5216718 | 6.51 | nM | Homo sapiens | ||
14. | ALA5218639 | (rac)-30a; VU6029053 | Activity | 0 | ALA5216717 | NA | Homo sapiens |