| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5218950 | 29f; VU6027634 | Papp | = | 0.374 | 10^-6 cm/s | ALA5216734 | 10^-6 cm/s | ||||
| 2. | ALA5218950 | 29f; VU6027634 | Ratio | = | 110 | ALA5216733 | ||||||
| 3. | ALA5218950 | 29f; VU6027634 | beta t1/2 | = | 86 | min | ALA5216732 | hr | ||||
| 4. | ALA5218950 | 29f; VU6027634 | Vdss | = | 0.61 | L/Kg | ALA5216731 | L.kg-1 | ||||
| 5. | ALA5218950 | 29f; VU6027634 | CL | = | 11.1 | ml/min.kg | ALA5216730 | mL.min-1.kg-1 | ||||
| 6. | ALA5218950 | 29f; VU6027634 | Fu | = | 0.2 | ALA5216729 | ||||||
| 7. | ALA5218950 | 29f; VU6027634 | Fu | = | 0.14 | ALA5216728 | ||||||
| 8. | ALA5218950 | 29f; VU6027634 | Fu | = | 0.03 | ALA5216727 | ||||||
| 9. | ALA5218950 | 29f; VU6027634 | Activity | = | 50 | % | ALA5216726 | % | Homo sapiens | |||
| 10. | ALA5218950 | 29f; VU6027634 | IC50 | > | 10000 | nM | ALA5216725 | nM | Homo sapiens | |||
| 11. | ALA5218950 | 29f; VU6027634 | IC50 | > | 10000 | nM | ALA5216724 | nM | Rattus norvegicus | |||
| 12. | ALA5218950 | 29f; VU6027634 | Activity | = | 4 | % | ALA5216723 | % | Rattus norvegicus | |||
| 13. | ALA5218950 | 29f; VU6027634 | IC50 | = | 1330 | nM | ALA5216722 | 5.88 | nM | Rattus norvegicus | ||
| 14. | ALA5218950 | 29f; VU6027634 | CL | = | 45 | ml/min.kg | ALA5216721 | mL.min-1.kg-1 | ||||
| 15. | ALA5218950 | 29f; VU6027634 | CL | = | 5 | ml/min.kg | ALA5216720 | mL.min-1.kg-1 | ||||
| 16. | ALA5218950 | 29f; VU6027634 | Activity | = | 2 | % | ALA5216719 | % | Homo sapiens | |||
| 17. | ALA5218950 | 29f; VU6027634 | IC50 | = | 304 | nM | ALA5216718 | 6.52 | nM | Homo sapiens | ||
| 18. | ALA5218950 | 29f; VU6027634 | Activity | 0 | ALA5216717 | NA | Homo sapiens | |||||
| 19. | ALA5218950 | 29f; VU6027634 | Activity | = | 35 | % | ALA5216716 | % | Rattus norvegicus |
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