# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5219602 | 41 | Fu | = | 0.47 | % | ALA5218193 | |||||
2. | ALA5219602 | 41 | Fu | = | 0.68 | % | ALA5218191 | |||||
3. | ALA5219602 | 41 | pKd | = | 5.9 | ALA5218190 | 5.90 | nM | Homo sapiens | |||
4. | ALA5219602 | 41 | t1/2 | > | 1000 | hr | ALA5218189 | hr | ||||
5. | ALA5219602 | 41 | t1/2 | = | 1.4 | hr | ALA5218188 | hr | ||||
6. | ALA5219602 | 41 | Vduss | = | 5.7 | L/Kg | ALA5218187 | L.kg-1 | ||||
7. | ALA5219602 | 41 | Vdss | = | 2.7 | L/Kg | ALA5218186 | L.kg-1 | ||||
8. | ALA5219602 | 41 | CL free | = | 60 | ml/min.kg | ALA5218185 | mL.min-1.kg-1 | ||||
9. | ALA5219602 | 41 | CL | = | 28 | ml/min.kg | ALA5218184 | mL.min-1.kg-1 | ||||
10. | ALA5219602 | 41 | F | = | 79 | % | ALA5218183 | % | ||||
11. | ALA5219602 | 41 | F | = | 67 | % | ALA5218177 | % | ||||
12. | ALA5219602 | 41 | t1/2 | = | 0.74 | hr | ALA5218176 | hr | ||||
13. | ALA5219602 | 41 | Vduss | = | 1.9 | L/Kg | ALA5218175 | L.kg-1 | ||||
14. | ALA5219602 | 41 | Vdss | = | 1.3 | L/Kg | ALA5218174 | L.kg-1 | ||||
15. | ALA5219602 | 41 | CL free | = | 38 | ml/min.kg | ALA5218173 | mL.min-1.kg-1 | ||||
16. | ALA5219602 | 41 | CL | = | 26 | ml/min.kg | ALA5218172 | mL.min-1.kg-1 | ||||
17. | ALA5219602 | 41 | CLH | < | 0.45 | ml/min/g | ALA5218160 | mL.min-1.g-1 | ||||
18. | ALA5219602 | 41 | CLH | < | 0.65 | ml/min/g | ALA5218159 | mL.min-1.g-1 | ||||
19. | ALA5219602 | 41 | CLH | < | 0.8 | ml/min/g | ALA5218158 | mL.min-1.g-1 | ||||
20. | ALA5219602 | 41 | solubility | > | 1000 | ug ml-1 | ALA5218157 | ug.mL-1 |