# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5220371 | 12a | Activity | 0 | ALA5217335 | Active | Mus musculus | |||||
2. | ALA5220371 | 12a | Ki | = | 36 | nM | ALA5217334 | 7.44 | nM | |||
3. | ALA5220371 | 12a | INH | = | 86.5 | % | ALA5217333 | % | ||||
4. | ALA5220371 | 12a | INH | = | 82 | % | ALA5217332 | % | ||||
5. | ALA5220371 | 12a | INH | < | 75 | % | ALA5217331 | % | Homo sapiens | |||
6. | ALA5220371 | 12a | INH | < | 75 | % | ALA5217330 | % | Homo sapiens | |||
7. | ALA5220371 | 12a | INH | < | 75 | % | ALA5217329 | % | Homo sapiens | |||
8. | ALA5220371 | 12a | INH | < | 75 | % | ALA5217328 | % | Homo sapiens | |||
9. | ALA5220371 | 12a | Ki | = | 0.069 | nM | ALA5217327 | 10.16 | nM | Homo sapiens | ||
10. | ALA5220371 | 12a | IC50 | = | 8.2 | nM | ALA5217326 | 8.09 | nM | Rattus norvegicus | ||
11. | ALA5220371 | 12a | CLH | = | 22.49 | microL/min/mg | ALA5217325 | mL.min-1.g-1 | ||||
12. | ALA5220371 | 12a | t1/2 | = | 61.63 | min | ALA5217324 | hr | ||||
13. | ALA5220371 | 12a | CLH | = | 51.82 | microL/min/mg | ALA5217323 | mL.min-1.g-1 | ||||
14. | ALA5220371 | 12a | t1/2 | = | 26.75 | min | ALA5217322 | hr | ||||
15. | ALA5220371 | 12a | INH | = | 99 | % | ALA5217321 | % | Homo sapiens | |||
16. | ALA5220371 | 12a | INH | = | 101 | % | ALA5217320 | % | Rattus norvegicus | |||
17. | ALA5220371 | 12a | INH | < | 75 | % | ALA5217319 | % | Homo sapiens | |||
18. | ALA5220371 | 12a | Ki | = | 150 | nM | ALA5217318 | 6.82 | nM | |||
19. | ALA5220371 | 12a | Activity | = | 34 | % | ALA5217316 | % | Mus musculus | |||
20. | ALA5220371 | 12a | Activity | = | 24 | % | ALA5217315 | % | Mus musculus |