# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5220590 | 38 | Activity | 0 | ALA5217974 | Non-Toxic | ||||||
2. | ALA5220590 | 38 | Km | = | 20.17 | uM | ALA5217973 | nM | Homo sapiens | |||
3. | ALA5220590 | 38 | Km | = | 13.88 | uM | ALA5217972 | nM | Homo sapiens | |||
4. | ALA5220590 | 38 | Ratio | = | 0.79 | ALA5217969 | Homo sapiens | |||||
5. | ALA5220590 | 38 | Activity | 0 | ALA5217968 | Non-Toxic | ||||||
6. | ALA5220590 | 38 | Activity | 0 | ALA5217967 | NA | ||||||
7. | ALA5220590 | 38 | Activity | 0 | ALA5217966 | Active | ||||||
8. | ALA5220590 | 38 | Activity | 0 | ALA5217965 | Active | ||||||
9. | ALA5220590 | 38 | Activity | 0 | ALA5217964 | Active | ||||||
10. | ALA5220590 | 38 | Activity | 0 | ALA5217963 | Active | ||||||
11. | ALA5220590 | 38 | PPB | < | 24 | % | ALA5217961 | % | ||||
12. | ALA5220590 | 38 | PPB | < | 38 | % | ALA5217960 | % | ||||
13. | ALA5220590 | 38 | IC50 | > | 30 | uM | ALA5217959 | nM | Homo sapiens | |||
14. | ALA5220590 | 38 | Vdss | = | 0.877 | L/Kg | ALA5217958 | L.kg-1 | ||||
15. | ALA5220590 | 38 | solubility | >= | 50 | ug ml-1 | ALA5217957 | ug.mL-1 | ||||
16. | ALA5220590 | 38 | Papp | = | 21.77 | 10^-6 cm/s | ALA5217956 | 10^-6 cm/s | ||||
17. | ALA5220590 | 38 | Papp | = | 27.5 | 10^-6 cm/s | ALA5217955 | 10^-6 cm/s | ||||
18. | ALA5220590 | 38 | IC50 | > | 100 | uM | ALA5217954 | nM | Homo sapiens | |||
19. | ALA5220590 | 38 | F | = | 220 | % | ALA5217953 | % | ||||
20. | ALA5220590 | 38 | CL | = | 36.1 | ml/min.kg | ALA5217952 | mL.min-1.kg-1 |