# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5220715 | 51 | F | = | 20 | % | ALA5215563 | % | ||||
2. | ALA5220715 | 51 | Cp | = | 0.009 | uM | ALA5215562 | uM | ||||
3. | ALA5220715 | 51 | Cmax | = | 2.1 | uM | ALA5215561 | nM | ||||
4. | ALA5220715 | 51 | Tmax | = | 3 | hr | ALA5215560 | hr | ||||
5. | ALA5220715 | 51 | AUC | = | 9.7 | uM.hr | ALA5215559 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
6. | ALA5220715 | 51 | CL | = | 6 | ml/min.kg | ALA5215558 | mL.min-1.kg-1 | ||||
7. | ALA5220715 | 51 | t1/2 | = | 3.9 | hr | ALA5215557 | hr | ||||
8. | ALA5220715 | 51 | IC50 | = | 12 | uM | ALA5215556 | 4.92 | nM | Homo sapiens | ||
9. | ALA5220715 | 51 | EC50 | = | 78 | nM | ALA5215555 | 7.11 | nM | |||
10. | ALA5220715 | 51 | EC50 | = | 91 | nM | ALA5215554 | 7.04 | nM | |||
11. | ALA5220715 | 51 | IC50 | = | 7600 | nM | ALA5215553 | 5.12 | nM | Homo sapiens | ||
12. | ALA5220715 | 51 | IC50 | = | 83 | nM | ALA5215552 | 7.08 | nM | Homo sapiens | ||
13. | ALA5220715 | 51 | IC50 | < | 1.5 | nM | ALA5215551 | nM | Homo sapiens | |||
14. | ALA5220715 | 51 | IC50 | = | 2.2 | nM | ALA5215550 | 8.66 | nM | Homo sapiens | ||
15. | ALA5220715 | 51 | IC50 | < | 1.5 | nM | ALA5215549 | nM | Homo sapiens |