| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5220926 | 31 | F | = | 4.1 | % | ALA5215570 | % | ||||
| 2. | ALA5220926 | 31 | Cp | = | 0.001 | uM | ALA5215569 | uM | ||||
| 3. | ALA5220926 | 31 | Cmax | = | 0.026 | uM | ALA5215568 | nM | ||||
| 4. | ALA5220926 | 31 | Tmax | = | 1.3 | hr | ALA5215567 | hr | ||||
| 5. | ALA5220926 | 31 | AUC | = | 0.1 | uM.hr | ALA5215566 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 6. | ALA5220926 | 31 | CL | = | 24 | ml/min.kg | ALA5215565 | mL.min-1.kg-1 | ||||
| 7. | ALA5220926 | 31 | t1/2 | = | 19 | hr | ALA5215564 | hr | ||||
| 8. | ALA5220926 | 31 | F | = | 7.9 | % | ALA5215563 | % | ||||
| 9. | ALA5220926 | 31 | Cp | = | 0.003 | uM | ALA5215562 | uM | ||||
| 10. | ALA5220926 | 31 | Cmax | = | 0.097 | uM | ALA5215561 | nM | ||||
| 11. | ALA5220926 | 31 | Tmax | = | 2.1 | hr | ALA5215560 | hr | ||||
| 12. | ALA5220926 | 31 | AUC | = | 0.47 | uM.hr | ALA5215559 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 13. | ALA5220926 | 31 | CL | = | 51 | ml/min.kg | ALA5215558 | mL.min-1.kg-1 | ||||
| 14. | ALA5220926 | 31 | t1/2 | = | 13 | hr | ALA5215557 | hr | ||||
| 15. | ALA5220926 | 31 | IC50 | = | 42 | uM | ALA5215556 | 4.38 | nM | Homo sapiens | ||
| 16. | ALA5220926 | 31 | EC50 | = | 10 | nM | ALA5215555 | 8.00 | nM | |||
| 17. | ALA5220926 | 31 | EC50 | = | 6 | nM | ALA5215554 | 8.22 | nM | |||
| 18. | ALA5220926 | 31 | IC50 | = | 6300 | nM | ALA5215553 | 5.20 | nM | Homo sapiens | ||
| 19. | ALA5220926 | 31 | IC50 | = | 350 | nM | ALA5215552 | 6.46 | nM | Homo sapiens | ||
| 20. | ALA5220926 | 31 | IC50 | < | 0.3 | nM | ALA5215551 | nM | Homo sapiens |
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