| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5220994 | 28 | INH | 0 | ALA5218028 | NA | % | Homo sapiens | ||||
| 2. | ALA5220994 | 28 | INH | 0 | ALA5218027 | Active | % | Homo sapiens | ||||
| 3. | ALA5220994 | 28 | INH | 0 | ALA5218026 | Active | % | Homo sapiens | ||||
| 4. | ALA5220994 | 28 | INH | 0 | ALA5218025 | NA | % | Homo sapiens | ||||
| 5. | ALA5220994 | 28 | INH | 0 | ALA5218024 | NA | % | Homo sapiens | ||||
| 6. | ALA5220994 | 28 | INH | 0 | ALA5218023 | NA | % | Homo sapiens | ||||
| 7. | ALA5220994 | 28 | INH | 0 | ALA5218022 | NA | % | Homo sapiens | ||||
| 8. | ALA5220994 | 28 | INH | 0 | ALA5218021 | NA | % | Homo sapiens | ||||
| 9. | ALA5220994 | 28 | INH | = | 80 | % | ALA5218020 | % | Homo sapiens | |||
| 10. | ALA5220994 | 28 | INH | = | 97 | % | ALA5218019 | % | Homo sapiens | |||
| 11. | ALA5220994 | 28 | MRT | = | 0.37 | hr | ALA5218016 | hr | ||||
| 12. | ALA5220994 | 28 | t1/2 | = | 0.3 | hr | ALA5218015 | hr | ||||
| 13. | ALA5220994 | 28 | Vdss | = | 2 | L/Kg | ALA5218014 | L.kg-1 | ||||
| 14. | ALA5220994 | 28 | CL | = | 95 | ml/min.kg | ALA5218013 | mL.min-1.kg-1 | ||||
| 15. | ALA5220994 | 28 | AUC | = | 102 | hr.ng/ml | ALA5218012 | ng.hr.mL-1 | ||||
| 16. | ALA5220994 | 28 | Cmax | = | 210 | ng/ml | ALA5218011 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 17. | ALA5220994 | 28 | Stability | > | 98 | % | ALA5217998 | % | ||||
| 18. | ALA5220994 | 28 | logD | = | 4.4 | ALA5217997 | ||||||
| 19. | ALA5220994 | 28 | pEC50 | = | 8.5 | ALA5217996 | 8.50 | nM | Homo sapiens | |||
| 20. | ALA5220994 | 28 | pIC50 | = | 10.1 | ALA5217994 | 10.10 | nM | Homo sapiens |
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