# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5266817 | 50 | INH | = | 52.9 | % | ALA5240435 | % | ||||
2. | ALA5266817 | 50 | QH | = | 31 | % | ALA5240429 | % | ||||
3. | ALA5266817 | 50 | t1/2 | = | 0.9 | hr | ALA5240428 | hr | ||||
4. | ALA5266817 | 50 | Vdss | = | 1.1 | L/Kg | ALA5240427 | L.kg-1 | ||||
5. | ALA5266817 | 50 | AUC | = | 1527 | mg.hr/ml | ALA5240426 | ng.hr.mL-1 | ||||
6. | ALA5266817 | 50 | CL | = | 17 | ml/min.kg | ALA5240425 | mL.min-1.kg-1 | ||||
7. | ALA5266817 | 50 | F | = | 34 | % | ALA5240424 | % | ||||
8. | ALA5266817 | 50 | Tmax | = | 0.87 | hr | ALA5240423 | hr | ||||
9. | ALA5266817 | 50 | Cmax | = | 894 | mg/ml | ALA5240422 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
10. | ALA5266817 | 50 | AUC | = | 2767 | mg.hr/ml | ALA5240421 | ng.hr.mL-1 | ||||
11. | ALA5266817 | 50 | INH | 0 | ALA5240419 | Not Active | % | Homo sapiens | ||||
12. | ALA5266817 | 50 | INH | 0 | ALA5240418 | Not Active | % | Homo sapiens | ||||
13. | ALA5266817 | 50 | INH | 0 | ALA5240417 | Not Active | % | Homo sapiens | ||||
14. | ALA5266817 | 50 | INH | 0 | ALA5240416 | Not Active | % | Homo sapiens | ||||
15. | ALA5266817 | 50 | INH | 0 | ALA5240415 | Not Active | % | Homo sapiens | ||||
16. | ALA5266817 | 50 | INH | 0 | ALA5240414 | Not Active | % | Homo sapiens | ||||
17. | ALA5266817 | 50 | IC50 | > | 10 | uM | ALA5240413 | nM | Homo sapiens | |||
18. | ALA5266817 | 50 | IC50 | > | 10 | uM | ALA5240412 | nM | Homo sapiens | |||
19. | ALA5266817 | 50 | IC50 | > | 10 | uM | ALA5240411 | nM | Homo sapiens | |||
20. | ALA5266817 | 50 | IC50 | > | 10 | uM | ALA5240410 | nM | Homo sapiens |