# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5267355 | GJ2 | Stability | 0 | ALA5225757 | Stable | % | |||||
2. | ALA5267355 | GJ2 | Kd | <= | 1 | 10^-12M | ALA5225755 | 10^-12M | Homo sapiens | |||
3. | ALA5267355 | GJ2 | INH | 0 | ALA5225754 | Dose-Dependent Effect | % | |||||
4. | ALA5267355 | GJ2 | INH | 0 | ALA5225753 | Active | % | Homo sapiens | ||||
5. | ALA5267355 | GJ2 | INH | 0 | ALA5225752 | Not Active | % | |||||
6. | ALA5267355 | GJ2 | INH | = | 100 | % | ALA5225751 | % | Homo sapiens | |||
7. | ALA5267355 | GJ2 | Activity | 0 | ALA5225750 | Not Active | ||||||
8. | ALA5267355 | GJ2 | INH | 0 | ALA5225749 | Not Active | % | Bos taurus | ||||
9. | ALA5267355 | GJ2 | IC50 | = | 0.05 | uM | ALA5225748 | 7.30 | nM | Homo sapiens | ||
10. | ALA5267355 | GJ2 | Activity | 0 | ALA5225747 | Active | Homo sapiens | |||||
11. | ALA5267355 | GJ2 | INH | 0 | ALA5225746 | Dose-Dependent Effect | % | Homo sapiens | ||||
12. | ALA5267355 | GJ2 | Activity | = | 6.3 | % | ALA5225745 | % | Homo sapiens | |||
13. | ALA5267355 | GJ2 | Activity | = | 10 | % | ALA5225744 | % | Homo sapiens | |||
14. | ALA5267355 | GJ2 | Activity | = | 14.3 | % | ALA5225743 | % | Homo sapiens | |||
15. | ALA5267355 | GJ2 | CL | = | 19.63 | L/hr/kg | ALA5225740 | mL.min-1.kg-1 | ||||
16. | ALA5267355 | GJ2 | t1/2 | = | 4.89 | hr | ALA5225739 | hr | ||||
17. | ALA5267355 | GJ2 | Stability | = | 74 | % | ALA5225738 | % |