| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5267404 | 12 | IC50 | > | 25 | uM | ALA5225644 | nM | Homo sapiens | |||
| 2. | ALA5267404 | 12 | F | = | 7 | % | ALA5225637 | % | ||||
| 3. | ALA5267404 | 12 | CLH | < | 0.5 | L/hr/kg | ALA5225636 | mL.min-1.kg-1 | ||||
| 4. | ALA5267404 | 12 | IC50 | = | 91 | nM | ALA5225635 | 7.04 | nM | Homo sapiens | ||
| 5. | ALA5267404 | 12 | Ki | = | 2.7 | nM | ALA5225634 | 8.57 | nM | Homo sapiens | ||
| 6. | ALA5267404 | 12 | permeability | = | 1.1 | 10^-6 cm/s | ALA5225633 | 10^-6 cm/s | ||||
| 7. | ALA5267404 | 12 | IC50 | > | 25 | uM | ALA5225632 | nM | Homo sapiens | |||
| 8. | ALA5267404 | 12 | IC50 | = | 1624 | nM | ALA5225631 | 5.79 | nM | Homo sapiens | ||
| 9. | ALA5267404 | 12 | IC50 | = | 1507 | nM | ALA5225630 | 5.82 | nM | Homo sapiens | ||
| 10. | ALA5267404 | 12 | IC50 | = | 7471 | nM | ALA5225629 | 5.13 | nM | Homo sapiens | ||
| 11. | ALA5267404 | 12 | INH | 0 | ALA5225628 | Tde | % | Homo sapiens | ||||
| 12. | ALA5267404 | 12 | Fu | = | 41 | % | ALA5225627 | |||||
| 13. | ALA5267404 | 12 | CL | = | 7.1 | L/hr/kg | ALA5225626 | mL.min-1.kg-1 | ||||
| 14. | ALA5267404 | 12 | AUC | = | 456 | nM.hr | ALA5225625 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 15. | ALA5267404 | 12 | CL | = | 1.2 | L/hr/kg | ALA5225624 | mL.min-1.kg-1 | ||||
| 16. | ALA5267404 | 12 | t1/2 | = | 5.5 | hr | ALA5225623 | hr | ||||
| 17. | ALA5267404 | 12 | Vdss | = | 4.6 | L/hr/kg | ALA5225622 | L/hr/kg | ||||
| 18. | ALA5267404 | 12 | AUC | = | 759 | nM.hr | ALA5225621 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | ng.hr.mL-1 |
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