# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5268293 | 12 | Activity | = | 33.5 | % | ALA5250924 | % | ||||
2. | ALA5268293 | 12 | CLH | = | 3 | ml/min/g | ALA5250914 | mL.min-1.g-1 | ||||
3. | ALA5268293 | 12 | CLH | = | 10.2 | ml/min/g | ALA5250913 | mL.min-1.g-1 | ||||
4. | ALA5268293 | 12 | CLH | = | 11.4 | ml/min/g | ALA5250912 | mL.min-1.g-1 | ||||
5. | ALA5268293 | 12 | t1/2 | = | 693 | min | ALA5250909 | hr | ||||
6. | ALA5268293 | 12 | t1/2 | = | 206 | min | ALA5250908 | hr | ||||
7. | ALA5268293 | 12 | t1/2 | = | 184 | min | ALA5250907 | hr | ||||
8. | ALA5268293 | 12 | AUClast | = | 25981 | hr.ng/ml | ALA5250906 | ng.hr.mL-1 | ||||
9. | ALA5268293 | 12 | Cmax | = | 2170 | ng/ml | ALA5250905 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
10. | ALA5268293 | 12 | Tmax | = | 3 | hr | ALA5250904 | hr | ||||
11. | ALA5268293 | 12 | t1/2 | = | 7 | hr | ALA5250903 | hr | ||||
12. | ALA5268293 | 12 | Ratio | = | 6 | ALA5250902 | ||||||
13. | ALA5268293 | 12 | EC50 | = | 0.2 | uM | ALA5250901 | 6.70 | nM | Homo sapiens | ||
14. | ALA5268293 | 12 | EC50 | = | 0.74 | uM | ALA5250900 | 6.13 | nM | Homo sapiens |