# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5268479 | 1bj | PB | = | 87 | % | ALA5265280 | % | Homo sapiens | |||
2. | ALA5268479 | 1bj | Papp | = | 220 | nm/s | ALA5265279 | nm/s | ||||
3. | ALA5268479 | 1bj | solubility | = | 0.031 | mg/ml | ALA5265278 | ug.mL-1 | ||||
4. | ALA5268479 | 1bj | AUC/dose | = | 152 | ng/hr/ml | ALA5265277 | ng/hr/ml | ||||
5. | ALA5268479 | 1bj | t1/2 | > | 180 | min | ALA5265276 | hr | ||||
6. | ALA5268479 | 1bj | EC50 | = | 54 | nM | ALA5265274 | 7.27 | nM | Rattus norvegicus | ||
7. | ALA5268479 | 1bj | IC50 | = | 7.1 | nM | ALA5265273 | 8.15 | nM | Homo sapiens |