# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5269176 | 17k | Stability | 0 | ALA5231947 | Not Determined | % | |||||
2. | ALA5269176 | 17k | Stability | = | 96 | % | ALA5231946 | % | ||||
3. | ALA5269176 | 17k | Stability | 0 | ALA5231945 | Not Determined | % | |||||
4. | ALA5269176 | 17k | Stability | = | 8.5 | % | ALA5231944 | % | ||||
5. | ALA5269176 | 17k | PPB | = | 74 | % | ALA5231943 | % | ||||
6. | ALA5269176 | 17k | PPB | = | 78 | % | ALA5231942 | % | ||||
7. | ALA5269176 | 17k | MIC | > | 32 | ug ml-1 | ALA5231941 | ug.mL-1 | Cryptococcus neoformans | |||
8. | ALA5269176 | 17k | MIC | > | 32 | ug ml-1 | ALA5231940 | ug.mL-1 | Candida albicans | |||
9. | ALA5269176 | 17k | MIC | > | 32 | ug ml-1 | ALA5231939 | ug.mL-1 | Pseudomonas aeruginosa | |||
10. | ALA5269176 | 17k | MIC | > | 32 | ug ml-1 | ALA5231938 | ug.mL-1 | Acinetobacter baumannii | |||
11. | ALA5269176 | 17k | MIC | > | 32 | ug ml-1 | ALA5231937 | ug.mL-1 | Klebsiella pneumoniae | |||
12. | ALA5269176 | 17k | MIC | > | 32 | ug ml-1 | ALA5231936 | ug.mL-1 | Escherichia coli | |||
13. | ALA5269176 | 17k | MIC | > | 32 | ug ml-1 | ALA5231935 | ug.mL-1 | Staphylococcus aureus | |||
14. | ALA5269176 | 17k | IC50 | > | 50 | uM | ALA5231934 | nM | Entamoeba histolytica | |||
15. | ALA5269176 | 17k | IC50 | > | 23 | uM | ALA5231933 | nM | Giardia intestinalis | |||
16. | ALA5269176 | 17k | Activity | = | 86 | % | ALA5231925 | % | Trypanosoma brucei brucei | |||
17. | ALA5269176 | 17k | CC50 | > | 100 | uM | ALA5231921 | nM | Homo sapiens | |||
18. | ALA5269176 | 17k | IC50 | = | 2.3 | uM | ALA5231920 | 5.64 | nM | Trypanosoma cruzi | ||
19. | ALA5269176 | 17k | MIC90 | > | 32 | ug ml-1 | ALA5231918 | ug.mL-1 | Mycobacterium tuberculosis | |||
20. | ALA5269176 | 17k | MIC90 | = | 16 | ug ml-1 | ALA5231917 | ug.mL-1 | Mycobacterium tuberculosis |