# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5271406 | 12; OFH611 | Activity | 0 | ALA5239865 | Not Active | Homo sapiens | |||||
2. | ALA5271406 | 12; OFH611 | Activity | 0 | ALA5239864 | Not Active | Homo sapiens | |||||
3. | ALA5271406 | 12; OFH611 | Activity | 0 | ALA5239863 | Active | Homo sapiens | |||||
4. | ALA5271406 | 12; OFH611 | Activity | 0 | ALA5239862 | Active | Homo sapiens | |||||
5. | ALA5271406 | 12; OFH611 | pKi | = | 9.84 | ALA5239861 | 9.84 | nM | Homo sapiens | |||
6. | ALA5271406 | 12; OFH611 | Ki | = | 0.14 | nM | ALA5239861 | 9.85 | nM | Homo sapiens | ||
7. | ALA5271406 | 12; OFH611 | pKi | = | 8.67 | ALA5239860 | 8.67 | nM | Homo sapiens | |||
8. | ALA5271406 | 12; OFH611 | Ki | = | 2.4 | nM | ALA5239860 | 8.62 | nM | Homo sapiens | ||
9. | ALA5271406 | 12; OFH611 | Activity | 0 | ALA5239859 | Non-Toxic | Cricetulus griseus | |||||
10. | ALA5271406 | 12; OFH611 | Kdiss | = | 0.026 | /min | ALA5239857 | /min | Homo sapiens | |||
11. | ALA5271406 | 12; OFH611 | ka | = | 0.09 | /min | ALA5239855 | /min | Homo sapiens | |||
12. | ALA5271406 | 12; OFH611 | Kd | = | 6 | nM | ALA5239854 | 8.22 | nM | Homo sapiens | ||
13. | ALA5271406 | 12; OFH611 | Kd | = | 6.5 | nM | ALA5239853 | 8.19 | nM | Homo sapiens | ||
14. | ALA5271406 | 12; OFH611 | Kd | = | 49.7 | nM | ALA5239852 | 7.30 | nM | Homo sapiens | ||
15. | ALA5271406 | 12; OFH611 | Kd | = | 54 | nM | ALA5239851 | 7.27 | nM | Homo sapiens | ||
16. | ALA5271406 | 12; OFH611 | IC50 | = | 450 | nM | ALA5239848 | 6.35 | nM | Homo sapiens | ||
17. | ALA5271406 | 12; OFH611 | IC50 | = | 300 | nM | ALA5239847 | 6.52 | nM | Homo sapiens | ||
18. | ALA5271406 | 12; OFH611 | Selectivity ratio | = | 0.39 | ALA5239846 | ||||||
19. | ALA5271406 | 12; OFH611 | Selectivity ratio | = | 0.06 | ALA5239845 | ||||||
20. | ALA5271406 | 12; OFH611 | Selectivity ratio | = | 0.69 | ALA5239844 | Homo sapiens |