| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5271855 | 1q | t1/2 | > | 180 | min | ALA5265416 | hr | ||||
| 2. | ALA5271855 | 1q | BBR | = | 0.17 | ALA5265285 | ||||||
| 3. | ALA5271855 | 1q | F | = | 130 | % | ALA5265284 | % | ||||
| 4. | ALA5271855 | 1q | Vdss | = | 1.6 | L/Kg | ALA5265283 | L.kg-1 | ||||
| 5. | ALA5271855 | 1q | CL | = | 22 | ml/min.kg | ALA5265282 | mL.min-1.kg-1 | ||||
| 6. | ALA5271855 | 1q | beta t1/2 | = | 1.1 | hr | ALA5265281 | hr | ||||
| 7. | ALA5271855 | 1q | PB | = | 84 | % | ALA5265280 | % | Homo sapiens | |||
| 8. | ALA5271855 | 1q | Papp | = | 165 | nm/s | ALA5265279 | nm/s | ||||
| 9. | ALA5271855 | 1q | solubility | = | 0.027 | mg/ml | ALA5265278 | ug.mL-1 | ||||
| 10. | ALA5271855 | 1q | AUC/dose | = | 1040 | ng/hr/ml | ALA5265277 | ng/hr/ml | ||||
| 11. | ALA5271855 | 1q | EC50 | = | 94 | nM | ALA5265274 | 7.03 | nM | Rattus norvegicus | ||
| 12. | ALA5271855 | 1q | IC50 | = | 14 | nM | ALA5265273 | 7.85 | nM | Homo sapiens |
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