| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5271921 | 3 | Fa | > | 100 | % | ALA5256734 | % | ||||
| 2. | ALA5271921 | 3 | F | = | 54 | % | ALA5256733 | % | ||||
| 3. | ALA5271921 | 3 | Cmax | = | 143 | ng/ml | ALA5256732 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 4. | ALA5271921 | 3 | AUC | = | 709 | hr.ng/ml | ALA5256731 | ng.hr.mL-1 | ||||
| 5. | ALA5271921 | 3 | K(p,uu,brain) | = | 0.4 | ALA5256730 | ||||||
| 6. | ALA5271921 | 3 | Fu | = | 0.031 | ALA5256729 | ||||||
| 7. | ALA5271921 | 3 | AUC | = | 440 | hr.ng/ml | ALA5256728 | ng.hr.mL-1 | ||||
| 8. | ALA5271921 | 3 | t1/2 | = | 0.6 | hr | ALA5256727 | hr | ||||
| 9. | ALA5271921 | 3 | Vdss | = | 1.5 | L/Kg | ALA5256726 | L.kg-1 | ||||
| 10. | ALA5271921 | 3 | CL | = | 39 | ml/min.kg | ALA5256725 | mL.min-1.kg-1 | ||||
| 11. | ALA5271921 | 3 | logD | = | 4.9 | ALA5256723 | ||||||
| 12. | ALA5271921 | 3 | Kinetic_solubility | = | 10 | uM | ALA5256722 | nM | ||||
| 13. | ALA5271921 | 3 | Ratio | = | 1.1 | ALA5256721 | ||||||
| 14. | ALA5271921 | 3 | Papp | = | 46 | 10^-6 cm/s | ALA5256720 | 10^-6 cm/s | ||||
| 15. | ALA5271921 | 3 | CLH | < | 10 | microL/min/mg | ALA5256719 | mL.min-1.g-1 | ||||
| 16. | ALA5271921 | 3 | CLH | = | 46 | microL/min/mg | ALA5256718 | mL.min-1.g-1 | ||||
| 17. | ALA5271921 | 3 | pEC50 | = | 7.2 | ALA5256717 | 7.20 | nM | Homo sapiens |
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