| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5274220 | 12f; VU6029051 | Ratio | = | 32.3 | ALA5237949 | ||||||
| 2. | ALA5274220 | 12f; VU6029051 | Papp | = | 1.75 | 10^-6 cm/s | ALA5237948 | 10^-6 cm/s | ||||
| 3. | ALA5274220 | 12f; VU6029051 | Fu | = | 0.05 | ALA5237947 | ||||||
| 4. | ALA5274220 | 12f; VU6029051 | Fu | = | 0.03 | ALA5237946 | ||||||
| 5. | ALA5274220 | 12f; VU6029051 | Fu | = | 0.01 | ALA5237945 | ||||||
| 6. | ALA5274220 | 12f; VU6029051 | IC50 | > | 10000 | nM | ALA5237944 | nM | Homo sapiens | |||
| 7. | ALA5274220 | 12f; VU6029051 | Activity | = | 8 | % | ALA5237943 | % | Homo sapiens | |||
| 8. | ALA5274220 | 12f; VU6029051 | IC50 | > | 10000 | nM | ALA5237942 | nM | Homo sapiens | |||
| 9. | ALA5274220 | 12f; VU6029051 | Activity | = | 2 | % | ALA5237941 | % | Rattus norvegicus | |||
| 10. | ALA5274220 | 12f; VU6029051 | IC50 | = | 190 | nM | ALA5237940 | 6.72 | nM | Rattus norvegicus | ||
| 11. | ALA5274220 | 12f; VU6029051 | CL | = | 51 | ml/min.kg | ALA5237939 | mL.min-1.kg-1 | ||||
| 12. | ALA5274220 | 12f; VU6029051 | CL | = | 5 | ml/min.kg | ALA5237938 | mL.min-1.kg-1 | ||||
| 13. | ALA5274220 | 12f; VU6029051 | logD | = | 2.94 | ALA5237937 | ||||||
| 14. | ALA5274220 | 12f; VU6029051 | Activity | = | 2 | % | ALA5237936 | % | Homo sapiens | |||
| 15. | ALA5274220 | 12f; VU6029051 | IC50 | = | 87 | nM | ALA5237935 | 7.06 | nM | Homo sapiens |
The page will load shortly, Thanks for your patience!