# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5276719 | 2 | solubility | = | 247 | mg/L | ALA5243029 | ug.mL-1 | ||||
2. | ALA5276719 | 2 | IC50 | = | 5.5 | nM | ALA5243028 | 8.26 | nM | Homo sapiens | ||
3. | ALA5276719 | 2 | Fmax | = | 87 | % | ALA5243027 | % | ||||
4. | ALA5276719 | 2 | Fmax | = | 87 | % | ALA5243026 | % | ||||
5. | ALA5276719 | 2 | CLH | = | 0.5 | L/hr/kg | ALA5243025 | mL.min-1.kg-1 | ||||
6. | ALA5276719 | 2 | CLH | = | 0.5 | L/hr/kg | ALA5243024 | mL.min-1.kg-1 | ||||
7. | ALA5276719 | 2 | Papp | = | 239 | nm/s | ALA5243022 | nm/s | ||||
8. | ALA5276719 | 2 | Papp | = | 0 | nm/s | ALA5243021 | nm/s | ||||
9. | ALA5276719 | 2 | logD | = | 2.1 | ALA5243020 | ||||||
10. | ALA5276719 | 2 | IC50 | > | 50 | uM | ALA5243018 | nM | Homo sapiens | |||
11. | ALA5276719 | 2 | IC50 | = | 0.18 | uM | ALA5243017 | 6.75 | nM | Homo sapiens | ||
12. | ALA5276719 | 2 | IC50 | = | 0.059 | uM | ALA5243016 | 7.23 | nM | Homo sapiens | ||
13. | ALA5276719 | 2 | IC50 | = | 0.027 | uM | ALA5243015 | 7.57 | nM | Homo sapiens | ||
14. | ALA5276719 | 2 | IC50 | = | 0.005 | uM | ALA5243014 | 8.30 | nM | Homo sapiens |