# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5276728 | 3DM | Cp | 0 | ALA5236154 | Bld | ||||||
2. | ALA5276728 | 3DM | Ct | 0 | ALA5236153 | Bld | ||||||
3. | ALA5276728 | 3DM | Activity | 0 | ALA5236142 | Toxic | ||||||
4. | ALA5276728 | 3DM | Activity | 0 | ALA5236141 | Toxic | ||||||
5. | ALA5276728 | 3DM | Activity | 0 | ALA5236140 | Toxic | ||||||
6. | ALA5276728 | 3DM | Activity | 0 | ALA5236139 | Toxic | ||||||
7. | ALA5276728 | 3DM | Activity | 0 | ALA5236138 | Toxic | ||||||
8. | ALA5276728 | 3DM | Activity | 0 | ALA5236137 | Toxic | ||||||
9. | ALA5276728 | 3DM | LD50 | = | 74 | mg kg-1 | ALA5236136 | mg.kg-1 | ||||
10. | ALA5276728 | 3DM | LD50 | = | 48.4 | mg kg-1 | ALA5236135 | mg.kg-1 | ||||
11. | ALA5276728 | 3DM | Activity | = | 100 | % | ALA5236134 | % | ||||
12. | ALA5276728 | 3DM | Activity | 0 | ALA5236133 | Not Active | Mus musculus | |||||
13. | ALA5276728 | 3DM | ED50 | > | 100 | mg kg-1 | ALA5236049 | mg.kg-1 | Mus musculus | |||
14. | ALA5276728 | 3DM | IC50 | = | 1096 | nM | ALA5236048 | 5.96 | nM | Mus musculus | ||
15. | ALA5276728 | 3DM | Emax | = | 64 | % | ALA5236047 | % | Mus musculus | |||
16. | ALA5276728 | 3DM | EC50 | = | 166.1 | nM | ALA5236046 | 6.78 | nM | Mus musculus | ||
17. | ALA5276728 | 3DM | EC50 | = | 67.5 | nM | ALA5236041 | 7.17 | nM | Mus musculus | ||
18. | ALA5276728 | 3DM | Ki | = | 49.1 | nM | ALA5236040 | 7.31 | nM | Mus musculus | ||
19. | ALA5276728 | 3DM | Ki | = | 124.7 | nM | ALA5236039 | 6.90 | nM | Mus musculus | ||
20. | ALA5276728 | 3DM | Ki | = | 34.1 | nM | ALA5236038 | 7.47 | nM | Mus musculus |