# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5276884 | 18k | Activity | 0 | ALA5242469 | Not Active | Homo sapiens | |||||
2. | ALA5276884 | 18k | INH | 0 | ALA5242468 | Not Active | % | |||||
3. | ALA5276884 | 18k | Activity | 0 | ALA5242467 | Not Active | Homo sapiens | |||||
4. | ALA5276884 | 18k | Activity | 0 | ALA5242466 | Not Active | Homo sapiens | |||||
5. | ALA5276884 | 18k | INH | 0 | ALA5242465 | Not Active | % | |||||
6. | ALA5276884 | 18k | INH | 0 | ALA5242464 | Not Active | % | |||||
7. | ALA5276884 | 18k | Activity | 0 | ALA5242463 | Non-Toxic | ||||||
8. | ALA5276884 | 18k | Activity | 0 | ALA5242462 | Non-Toxic | ||||||
9. | ALA5276884 | 18k | T>IC50 | = | 4 | hr | ALA5242461 | hr | ||||
10. | ALA5276884 | 18k | F | = | 35 | % | ALA5242460 | % | ||||
11. | ALA5276884 | 18k | IC50 | = | 239 | nM | ALA5242457 | 6.62 | nM | Homo sapiens | ||
12. | ALA5276884 | 18k | IC50 | = | 137 | nM | ALA5242456 | 6.86 | nM | Homo sapiens | ||
13. | ALA5276884 | 18k | Ki | = | 11 | nM | ALA5242447 | 7.96 | nM | Homo sapiens | ||
14. | ALA5276884 | 18k | IC50 | = | 99 | nM | ALA5242447 | 7.00 | nM | Homo sapiens | ||
15. | ALA5276884 | 18k | Vdss | = | 0.6 | L/Kg | ALA5242446 | L.kg-1 | ||||
16. | ALA5276884 | 18k | CL | = | 0.6 | L/kg/hr | ALA5242445 | mL.min-1.kg-1 | ||||
17. | ALA5276884 | 18k | Ratio | = | 11 | ALA5242444 | ||||||
18. | ALA5276884 | 18k | solubility | = | 876 | ug ml-1 | ALA5242443 | ug.mL-1 | ||||
19. | ALA5276884 | 18k | CLH | = | 12 | uL/min | ALA5242442 | uL/min | ||||
20. | ALA5276884 | 18k | IC50 | = | 29 | uM | ALA5242438 | 4.54 | nM | Homo sapiens |