# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5278530 | 1n | t1/2 | > | 180 | min | ALA5265416 | hr | ||||
2. | ALA5278530 | 1n | PB | = | 73 | % | ALA5265280 | % | Homo sapiens | |||
3. | ALA5278530 | 1n | solubility | = | 0.013 | mg/ml | ALA5265278 | ug.mL-1 | ||||
4. | ALA5278530 | 1n | AUC/dose | = | 19.3 | ng/hr/ml | ALA5265277 | ng/hr/ml | ||||
5. | ALA5278530 | 1n | EC50 | = | 170 | nM | ALA5265274 | 6.77 | nM | Rattus norvegicus | ||
6. | ALA5278530 | 1n | IC50 | = | 12 | nM | ALA5265273 | 7.92 | nM | Homo sapiens |