| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5278881 | 9d | Drugexcretion | = | 1 | % | ALA5251577 | % | ||||
| 2. | ALA5278881 | 9d | CL free | = | 100 | ml/min.kg | ALA5251574 | mL.min-1.kg-1 | ||||
| 3. | ALA5278881 | 9d | CL | = | 22 | ml/min.kg | ALA5251573 | mL.min-1.kg-1 | ||||
| 4. | ALA5278881 | 9d | CL free | = | 710 | ml/min.kg | ALA5251572 | mL.min-1.kg-1 | ||||
| 5. | ALA5278881 | 9d | CL | = | 7.1 | ml/min.kg | ALA5251571 | mL.min-1.kg-1 | ||||
| 6. | ALA5278881 | 9d | CLH | = | 2.4 | microL/min/mg | ALA5251570 | mL.min-1.g-1 | ||||
| 7. | ALA5278881 | 9d | CLH | = | 2.8 | microL/min/mg | ALA5251569 | mL.min-1.g-1 | ||||
| 8. | ALA5278881 | 9d | CLH | < | 2 | microL/min/mg | ALA5251568 | mL.min-1.g-1 | ||||
| 9. | ALA5278881 | 9d | CLH | = | 16 | microL/min/mg | ALA5251567 | mL.min-1.g-1 | ||||
| 10. | ALA5278881 | 9d | CLH | = | 13 | microL/min/mg | ALA5251566 | mL.min-1.g-1 | ||||
| 11. | ALA5278881 | 9d | Fu | = | 22 | % | ALA5251565 | |||||
| 12. | ALA5278881 | 9d | Fu | = | 1 | % | ALA5251564 | |||||
| 13. | ALA5278881 | 9d | Fu | = | 11 | % | ALA5251563 | |||||
| 14. | ALA5278881 | 9d | logD | = | 3 | ALA5251562 | ||||||
| 15. | ALA5278881 | 9d | CLH | = | 1.18 | microL/min/mg | ALA5251561 | mL.min-1.g-1 | Homo sapiens | |||
| 16. | ALA5278881 | 9d | CLH | = | 0.41 | microL/min/mg | ALA5251560 | mL.min-1.g-1 | Homo sapiens | |||
| 17. | ALA5278881 | 9d | CLH | < | 10 | microL/min/mg | ALA5251559 | mL.min-1.g-1 | ||||
| 18. | ALA5278881 | 9d | IC50 | = | 21 | nM | ALA5251558 | 7.68 | nM | Homo sapiens | ||
| 19. | ALA5278881 | 9d | IC50 | = | 74.6 | nM | ALA5251557 | 7.13 | nM | Homo sapiens |
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